SCHEMBL4484839

SCHEMBL4484839

Cc1c(O)cc2c(c1C)N(c1cccc(O)c1)CC1(CCC1)C2

nearest known ligand 0.34

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
HSD17B10 Q99714 2/20 0.32
KDM4E B2RXH2 1/20 0.32
ALDH1A1 P00352 1/20 0.32
MAPT P10636 1/20 0.32
HPGD P15428 1/20 0.32
CASP1 P29466 1/20 0.32
CASP7 P55210 1/20 0.32
OPRD1 P41143 2/20 0.32
OPRK1 P41145 1/20 0.31
OPRM1 P35372 2/20 0.31
SIGMAR1 Q99720 1/20 0.31
FGFR1 P11362 1/20 0.30
DRD2 P14416 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4473362 0.86
SCHEMBL4463874 0.85 KMT2A (0.42) MEN1KMT2AHSD17B10KDM4EALDH1A1
SCHEMBL4463115 0.83 CYP11B2 (0.34)
SCHEMBL4472455 0.82 SPR (0.34) MEN1KMT2A
SCHEMBL4464111 0.82 SSTR5 (0.35)
SCHEMBL4472622 0.79 SSTR5 (0.39) MEN1KMT2AKDM4EALDH1A1MAPT
SCHEMBL4467896 0.78 KCNJ1 (0.39) OPRM1
SCHEMBL4481197 0.77 GRM5 (0.35)
SCHEMBL4473864 0.77 HSD17B10 (0.38) MEN1KMT2AHSD17B10ALDH1A1HPGD
SCHEMBL4468208 0.76 HSP90AA1 (0.35)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20060128790-A1 Spiro derivatives as lipoxygenase inhibitors GALILEO PHARMACEUTICALS, INC. 2006-06-15 US claimed
US-7576094-B2 Spiro derivatives as lipoxygenase inhibitors ELI LILLY AND COMPANY (US) 2009-08-18 US disclosed
US-7576094-B2 Spiro derivatives as lipoxygenase inhibitors ELI LILLY AND COMPANY (US) 2009-08-18 US disclosed
US-7576094-B2 Spiro derivatives as lipoxygenase inhibitors ELI LILLY AND COMPANY (US) 2009-08-18 US disclosed
US-20060128790-A1 Spiro derivatives as lipoxygenase inhibitors GALILEO PHARMACEUTICALS, INC. 2006-06-15 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060128790-A1 Spiro derivatives as lipoxygenase inhibitors ALOX15B, ALOX5, ALOX15 MEN1 4420/4885KMT2A 3967/4885HSD17B10 83/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.