Nordexfenfluramine

Nordexfenfluramine

SCHEMBL44927

CC(N)Cc1cccc(C(F)(F)F)c1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 2/20 1.00
HTR2B P41595 2/20 1.00
HTR2C P28335 1/20 1.00
SIGMAR1 Q99720 3/20 0.64
SLC6A4 P31645 2/20 0.64
LMNA P02545 1/20 0.64
MAPT P10636 1/20 0.64
ADRA2C P18825 1/20 0.64
ADRA1A P35348 1/20 0.64
DRD3 P35462 1/20 0.64
OPRK1 P41145 1/20 0.64
TAAR1 Q96RJ0 5/20 0.58
IDO1 P14902 2/20 0.56
TP53 P04637 1/20 0.55
CYP1A2 P05177 1/20 0.55
CYP3A4 P08684 1/20 0.55
CYP2D6 P10635 1/20 0.55
TSHR P16473 1/20 0.55
CYP2C19 P33261 1/20 0.55
PNMT P11086 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Nordexfenfluramine SCHEMBL29390405 1.00 HTR2A (1.00) HTR2AHTR2BHTR2CSIGMAR1SLC6A4
Nordexfenfluramine SCHEMBL4668266 1.00 HTR2A (1.00) HTR2AHTR2BHTR2CSIGMAR1SLC6A4
Nordexfenfluramine SCHEMBL30081494 1.00 HTR2A (1.00) HTR2AHTR2BHTR2CSIGMAR1SLC6A4
Nordexfenfluramine SCHEMBL30081489 1.00 HTR2A (1.00) HTR2AHTR2BHTR2CSIGMAR1SLC6A4
Nordexfenfluramine SCHEMBL895637 1.00 HTR2A (1.00) HTR2AHTR2BHTR2CSIGMAR1SLC6A4
Nordexfenfluramine SCHEMBL29538965 0.98 HTR2A (0.96) HTR2AHTR2BHTR2CSIGMAR1SLC6A4
Nordexfenfluramine SCHEMBL8412627 0.98 HTR2A (0.96) HTR2AHTR2BHTR2CSIGMAR1SLC6A4
Nordexfenfluramine SCHEMBL10562287 0.98 HTR2A (0.96) HTR2AHTR2BHTR2CSIGMAR1SLC6A4
Nordexfenfluramine SCHEMBL16673896 0.92 HTR2A (0.84) HTR2AHTR2BHTR2CSIGMAR1SLC6A4
Nordexfenfluramine SCHEMBL16673917 0.92 HTR2A (0.84) HTR2AHTR2BHTR2CSIGMAR1SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1213 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2026107229-A1 REDUCING THE ADDICTIVE LIABILITY OF OPIOID ANALGESICS BY CO- ADMINISTERING 5HT2 RECEPTOR AGONISTS THE BOARD OF TRUSTEES OF THE LELAND STANFORD JUNIOR UNIVERSITY (US) 2026-05-21 WO claimed
EP-4722714-A1 SIMULTANEOUS ANALYSIS OF FOOD-BORNE DOPING SUBSTANCES USING LIQUID CHROMATOGRAPHY-MASS SPECTROMETRY (VFD: VACCINE FOR FOODBORNE DOPING) Korea Institute of Science and Technology (KR) 2026-04-08 EP claimed
US-12558326-B2 Method for treating epilepsy XENON PHARMACEUTICALS INC. (CA) 2026-02-24 US claimed
US-20250360137-A1 ENHANCEMENT OF THE EFFICACY OF SEROTONERGIC PSYCHEDELIC DRUGS IN THE TREATMENT OR PREVENTION OF CERTAIN NEUROPSYCHIATRIC DISORDERS THROUGH INHIBITION OF TYPE-9 PHOSPHODIESTERASES FREEDOM BIOSCIENCES INC (US) 2025-11-27 US claimed
US-20250295611-A1 METHODS OF TREATING 5HT2A RECEPTOR-MEDIATED CONDITIONS TESSELLATE THERAPEUTICS INC (US) 2025-09-25 US claimed
EP-4618980-A1 ENHANCEMENT OF THE EFFICACY OF SEROTONERGIC PSYCHEDELIC DRUGS IN THE TREATMENT OR PREVENTION OF CERTAIN NEUROPSYCHIATRIC DISORDERS THROUGH INHIBITION OF TYPE-9 PHOSPHODIESTERASES Freedom Biosciences, Inc. (US) 2025-09-24 EP claimed
EP-3687576-B1 USE OF CANNABIDIOL IN COMBINATION WITH NORFENFLURAMINE OR FENFLURAMINE IN THE TREATMENT OF EPILEPSY JAZZ PHARMACEUTICALS RESEARCH UK LTD (GB) 2025-09-03 EP claimed
EP-3518975-B1 FORMULATION COMPRISING FENFLURAMINE AND CANNABIDIOL AND ITS USE IN THE TREATMENT OF SEIZURES ZOGENIX INTERNATIONAL LTD (GB) 2025-04-09 EP claimed
US-20250032503-A1 USE OF APREPITANT FOR TREATING ALZHEIMER'S DISEASE HOTH THERAPEUTICS, INC. 2025-01-30 US claimed
CN-118873517-A Use of cannabidiol in combination with a 5-HT2B receptor agonist 上海柯西医药科技发展有限公司 2024-11-01 CN claimed
EP-0875498-A2 Process for the production of the isomers (R) and (S)-Alpha-methyl-3-(trifluoromethyl)benzeneethanamine Alfa Chemicals Italiana S.r.l. (IT) 1998-11-04 EP claimed
US-5808156-A Process for the production of the isomers (R) and (S)-α-methyl-3(trifluoromethyl)benzeneethanamine ALFA CHEMICALS ITALIANA S.P.A. (IT) 1998-09-15 US claimed
EP-0441160-B1 Process for preparing levo and dextro fenfluramine LAB MAG SPA (IT) 1995-07-05 EP claimed
EP-0440704-A1 COMPOSITIONS FOR TREATING TOBACCO WITHDRAWEL SYMPTOMS. MASSACHUSETTS INST TECHNOLOGY (US) 1991-08-14 EP claimed
WO-1990004387-A2 COMPOSITIONS FOR TREATING TOBACCO WITHDRAWAL SYMPTOMS MASSACHUSETTS INSTITUTE OF TECHNOLOGY (US) 1990-05-03 WO claimed
EP-0302757-A2 Anti-emetic serotonin depleting agents A.H. ROBINS COMPANY, INCORPORATED (US) 1989-02-08 EP claimed
EP-0053175-A4 USE OF d-FENFLURAMINE FOR THE MANUFACTURE OF A MEDICAMENT FOR MODIFYING FEEDING BEHAVIOR. MASSACHUSETTS INST TECHNOLOGY (US) 1982-10-07 EP claimed
EP-0053175-A1 USE OF d-FENFLURAMINE FOR THE MANUFACTURE OF A MEDICAMENT FOR MODIFYING FEEDING BEHAVIOR. MASSACHUSETTS INST TECHNOLOGY (US) 1982-06-09 EP claimed
WO-1981003611-A1 METHOD AND COMPOSITION FOR UTILIZING D-FENFLURAMINE FOR MODIFYING FEEDING BEHAVIOR MASSACHUSETTS INST TECHNOLOGY (US) 1981-12-24 WO claimed
US-4115587-A TREATMENT OF ATHEROSCLEROSIS AND HYPERCHOLESTER-EMIA A. H. ROBINS COMPANY, INC. (US) 1978-09-19 US claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250360137-A1 ENHANCEMENT OF THE EFFICACY OF SEROTONERGIC PSYCHEDELIC DRUGS IN THE TREATMENT OR PREVENTION OF CERTAIN NEUROPSYCHIATRIC DISORDERS THROUGH INHIBITION OF TYPE-9 PHOSPHODIESTERASES PDE9A, PDE3A, PDE2A HTR2A 14/4885HTR2B 28/4885HTR2C 42/4885
US-20250032503-A1 USE OF APREPITANT FOR TREATING ALZHEIMER'S DISEASE TACR1, ACHE, TACR2 HTR2A 207/4885HTR2B 343/4885HTR2C 390/4885
US-20250295611-A1 METHODS OF TREATING 5HT2A RECEPTOR-MEDIATED CONDITIONS HTR2A, HTR5A, HTR6 HTR2A 1/4885HTR2B 7/4885HTR2C 5/4885
US-12558326-B2 Method for treating epilepsy PNMT, SLC6A1, CPT1B HTR2A 239/4885HTR2B 790/4885HTR2C 159/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.