Hydrochloric Acid

Hydrochloric Acid

SCHEMBL4496228

CN1CCC(Oc2cccc(NC(=O)c3ccncc3)n2)CC1.[Cl-].[H+]

nearest known ligand 0.53

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHEBDKRB2CHRM1CHRM2CHRM3CHRNA1CHRNB1CHRNDCHRNECHRNGGUCY1A1GUCY1A2GUCY1B1GUCY1B2NAMPTPTAFRSLC10A2SLC6A2SLC6A3TACR1dacAdacBdacCftsImrcAmrcBmrdA

The experimentally established mechanism targets of Hydrochloric Acid. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1F P30939 12/20 0.53
HTR1A P08908 6/20 0.53
HTR1D P28221 5/20 0.53
HTR1B P28222 4/20 0.53
WNT1 P04628 6/20 0.47
GSK3B P49841 6/20 0.47
DYRK1A Q13627 6/20 0.47
CLK2 P49760 1/20 0.43
CLK3 P49761 1/20 0.43
GRM5 P41594 1/20 0.42
HTR1E P28566 2/20 0.41
CHRM5 P08912 1/20 0.41
DRD5 P21918 1/20 0.41
HTR7 P34969 1/20 0.41
OPRK1 P41145 1/20 0.41
TMEM97 Q5BJF2 1/20 0.41
SIGMAR1 Q99720 1/20 0.41
HTR2A P28223 1/20 0.41
HTR2C P28335 1/20 0.41
HTR4 Q13639 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10267501 0.99 HTR1F (0.54) HTR1FHTR1AHTR1DHTR1BWNT1
Hydrochloric Acid SCHEMBL4496232 0.98 HTR1F (0.53) HTR1FHTR1AHTR1DHTR1BWNT1
Hydrochloric Acid SCHEMBL4510534 0.89 HTR1F (0.64) HTR1FHTR1AHTR1DHTR1BHTR1E
SCHEMBL10267497 0.87 HTR1F (0.67) HTR1FHTR1AHTR1DHTR1BHTR1E
Hydrochloric Acid SCHEMBL4498244 0.86 HTR1F (0.66) HTR1FHTR1AHTR1DHTR1BHTR1E
Hydrochloric Acid SCHEMBL4495848 0.85 HTR1F (0.49) HTR1FHTR1AHTR1DHTR1BWNT1
Hydrochloric Acid SCHEMBL4495915 0.84 HTR1F (0.55) HTR1FHTR1AHTR1DHTR1BWNT1
SCHEMBL13675079 0.83 HTR1F (0.51) HTR1FHTR1AHTR1DHTR1BWNT1
SCHEMBL4502036 0.83 MAPK8 (0.52) HTR1FHTR1AHTR1DHTR1BGRM5
Hydrochloric Acid SCHEMBL4509156 0.82 ALDH1A1 (0.52) HTR1FHTR1AHTR1DHTR1BWNT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1626958-B1 (PIPERIDINYLOXY)PHENYL, (PIPERIDINYLOXY)PYRIDINYL, (PIPERIDINYLSULFANYL)PHENYL AND (PIPERIDINYLSULFANYL)PYRIDINYL COMPOUNDS AS 5-HT 1F AGONISTS LILLY CO ELI (US) 2012-06-27 EP disclosed
US-7608629-B2 (Piperidinyloxy)phenyl, (piperidinyloxy)pyridinyl, (piperidinylsulfanyl)phenyl and (piperidinylsulfanyl)pyridinyl compounds as 5-HT1F agonists ELI LILLY AND COMPANY (US) 2009-10-27 US disclosed
US-20060211734-A1 (Piperidinyloxy)phenyl, (piperidinyloxy)pyridinyl, (piperidinylsulfanyl)phenyl and (piperidinylsulfanyl)pyridinyl compounds as 5-ht1f agonists ELILILLY AND COMPANY (US) 2006-09-21 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060211734-A1 (Piperidinyloxy)phenyl, (piperidinyloxy)pyridinyl, (piperidinylsulfanyl)phenyl and (piperidinylsulfanyl)pyridinyl compounds as 5-ht1f agonists HTR1A, HTR1F, HTR5A HTR1F 2/4885HTR1A 1/4885HTR1D 5/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.