SCHEMBL4500338

SCHEMBL4500338

Cc1cccc(NC(=O)N2CCOC(COc3ccccc3F)C2)n1

nearest known ligand 0.46

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PDK1 Q15118 2/20 0.46
NPC1 O15118 2/20 0.44
RAB9A P51151 2/20 0.44
MAPT P10636 1/20 0.44
OPRM1 P35372 1/20 0.42
FKBP1A P62942 1/20 0.41
CCR3 P51677 3/20 0.40
DRD4 P21917 1/20 0.39
TSHR P16473 1/20 0.39
NR1H4 Q96RI1 1/20 0.39
HRH3 Q9Y5N1 1/20 0.38
GRM5 P41594 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4506372 0.89 TRPV1 (0.43) PDK1MAPTFKBP1ACCR3DRD4
SCHEMBL4510657 0.89 PDK1 (0.46) PDK1NPC1RAB9AMAPTDRD4
SCHEMBL4498562 0.88 EPHA2 (0.44) PDK1OPRM1CCR3DRD4GRM5
Trifluoroacetic Acid SCHEMBL4495237 0.85 TRPV1 (0.40) PDK1CCR3DRD4NR1H4GRM5
SCHEMBL4509367 0.79 MEN1 (0.51) PDK1NPC1RAB9AMAPTDRD4
SCHEMBL4496536 0.78 RBP4 (0.46) PDK1
Trifluoroacetic Acid SCHEMBL4516194 0.78 GRM5 (0.40) PDK1CCR3DRD4TSHRGRM5
SCHEMBL4490668 0.78 EPHA2 (0.43) PDK1CCR3DRD4
SCHEMBL4516917 0.77 EPHA2 (0.44) MAPTDRD4GRM5
SCHEMBL4507600 0.77 PDK1 (0.42) PDK1CCR3DRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090325956-A1 Aromatic amine derivative and use thereof TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-12-31 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090325956-A1 Aromatic amine derivative and use thereof SCD, SCD5, SMS PDK1 663/4885NPC1 57/4885RAB9A 3368/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.