SCHEMBL4500980

SCHEMBL4500980

NC(=O)[CH]CN1CCN(c2cccc(N)n2)CC1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIN2D O15399 1/20 0.42
GRIN3B O60391 1/20 0.42
GRIN1 Q05586 1/20 0.42
GRIN2A Q12879 1/20 0.42
GRIN2B Q13224 1/20 0.42
GRIN2C Q14957 1/20 0.42
GRIN3A Q8TCU5 1/20 0.42
HTR1A P08908 5/20 0.36
HTR2A P28223 3/20 0.36
DRD3 P35462 3/20 0.36
ALDH1A1 P00352 1/20 0.36
NOS1 P29475 2/20 0.36
DRD2 P14416 1/20 0.36
DRD4 P21917 1/20 0.36
HTR2C P28335 1/20 0.36
HTR7 P34969 1/20 0.36
NOS3 P29474 1/20 0.35
AOC3 Q16853 2/20 0.35
PARP1 P09874 2/20 0.35
BDKRB1 P46663 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5452260 0.80 GRIN2D (0.46) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL4486164 0.80 HTR1A (0.55) HTR1AHTR2ADRD3ALDH1A1DRD2
SCHEMBL4498299 0.77 OGA (0.38) HTR1AALDH1A1AOC3
SCHEMBL31052529 0.76 GRIN2D (0.47) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL24322998 0.75 HRH3 (0.56) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL27913890 0.74 GRIN2D (0.48) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL4510839 0.73 SORD (0.49) HTR1ADRD2DRD4AOC3PARP1
SCHEMBL5452265 0.73 DRD2 (0.50) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL4327175 0.73 ALDH1A1 (0.49) HTR1AHTR2ADRD3ALDH1A1DRD2
SCHEMBL4704790 0.71 SMN1; SMN2 (0.51) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7491821-B2 2-(4-fluorophenyl)-4-propyl-oxazole-5-carboxylic acid {2-[4-(6-aminopyridin-2-yl)-piperazin-1-yl]-1-methyl-ethyl}amide; purinergic receptor antagonists, analgesics; urogenital, gastointestinal and respiratory system disorders ROCHE PALO ALTO LLC (US) 2009-02-17 US disclosed