SCHEMBL4498299

SCHEMBL4498299

NC(=O)[CH]CN1CCN(c2nccc(N)n2)CC1

nearest known ligand 0.40

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
OGA O60502 1/20 0.38
ALDH1A1 P00352 4/20 0.38
KDM4E B2RXH2 3/20 0.38
HTR1A P08908 3/20 0.38
NPSR1 Q6W5P4 1/20 0.38
AOC3 Q16853 2/20 0.38
KDM1A O60341 1/20 0.37
TSHR P16473 1/20 0.37
HTT P42858 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
PANK3 Q9H999 1/20 0.37
PTPN11 Q06124 1/20 0.36
MDM2 Q00987 1/20 0.36
ACHE P22303 3/20 0.36
TDP1 Q9NUW8 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15740608 0.85 OGA (0.42) OGAALDH1A1KDM4EHTR1ANPSR1
SCHEMBL4327175 0.83 ALDH1A1 (0.49) ALDH1A1KDM4EHTR1ANPSR1TSHR
SCHEMBL5458684 0.81 OGA (0.44) OGAALDH1A1KDM4EKDM1ATSHR
SCHEMBL4500980 0.77 GRIN2D (0.42) ALDH1A1HTR1AAOC3
SCHEMBL4945954 0.75 SLC6A7 (0.46) OGAALDH1A1KDM4EKDM1ATSHR
SCHEMBL6800518 0.73 ACHE (0.55) OGAKDM4EPTPN11ACHE
SCHEMBL5458689 0.73 ACHE (0.56) OGAPTPN11ACHE
SCHEMBL4486164 0.73 HTR1A (0.55) ALDH1A1KDM4EHTR1ANPSR1SMN1; SMN2
SCHEMBL15740759 0.72 KDM4E (0.49) ALDH1A1KDM4ENPSR1KDM1ASMN1; SMN2
SCHEMBL4510839 0.72 SORD (0.49) HTR1AAOC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7491821-B2 2-(4-fluorophenyl)-4-propyl-oxazole-5-carboxylic acid {2-[4-(6-aminopyridin-2-yl)-piperazin-1-yl]-1-methyl-ethyl}amide; purinergic receptor antagonists, analgesics; urogenital, gastointestinal and respiratory system disorders ROCHE PALO ALTO LLC (US) 2009-02-17 US disclosed