SCHEMBL45068

SCHEMBL45068

CN(C)CCNC(=O)Cc1nc(-c2cccc(-c3cn4ncccc4n3)c2)no1

nearest known ligand 0.41

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HPGD P15428 2/20 0.38
TSHR P16473 2/20 0.38
FYN P06241 4/20 0.37
HDAC4 P56524 1/20 0.36
HDAC1 Q13547 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36
KMT2A Q03164 1/20 0.36
CAMK2D Q13557 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
ALDH1A1 P00352 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL44594 0.92 HTR1A (0.39) HDAC4HDAC1HDAC6KMT2ACAMK2D
SCHEMBL44314 0.89 HDAC4 (0.42) HPGDHDAC4HDAC6ALDH1A1
SCHEMBL44565 0.88 HPGD (0.51) HPGDTSHRHDAC4HDAC6KMT2A
SCHEMBL44472 0.87 HTT (0.40) TSHRHDAC1KMT2A
SCHEMBL38209 0.86 GSK3B (0.43) FYNHDAC4HDAC1HDAC6CAMK2D
SCHEMBL994121 0.85 LMNA (0.46) TSHRKMT2AALDH1A1
SCHEMBL46482 0.82 FYN (0.34) FYNHDAC4HDAC1HDAC6CAMK2D
SCHEMBL44623 0.82 FFAR1 (0.42) TSHRKMT2AALDH1A1
SCHEMBL44354 0.82 HPGD (0.45) HPGDTSHRKMT2AALDH1A1
SCHEMBL45433 0.81 GLA (0.37) KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011137587-A1 CYTOKINE INHIBITORS HUTCHISON MEDIPHARMA LIMITED (CN) 2011-11-10 WO disclosed