SCHEMBL4510362

SCHEMBL4510362

CCCCCc1ccc2[nH]ccc(=O)c2c1

nearest known ligand 0.53

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 2/20 0.53
HTR1D P28221 1/20 0.53
HTR1B P28222 1/20 0.53
GPR84 Q9NQS5 1/20 0.46
GABRA1 P14867 3/20 0.44
GABRB2 P47870 3/20 0.44
CTSV O60911 2/20 0.44
CTSL P07711 2/20 0.44
GHSR Q92847 3/20 0.44
RORA P35398 1/20 0.41
RORC P51449 1/20 0.41
RORB Q92753 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2056367 0.82 GABRA1 (0.48) HTR1AHTR1DHTR1BGABRA1GABRB2
SCHEMBL7282642 0.80 ALDH1A1 (0.42) GABRA1GABRB2
SCHEMBL4531377 0.78 HTR1A (0.50) HTR1AHTR1DHTR1BGPR84GABRA1
SCHEMBL4531373 0.78 HTR1A (0.50) HTR1AHTR1DHTR1BGPR84GABRA1
SCHEMBL6629875 0.78 HDAC1 (0.57) HTR1AHTR1DHTR1BGPR84
SCHEMBL564963 0.76 HDAC1 (0.56) HTR1AHTR1DHTR1BGPR84
SCHEMBL20382323 0.75 GHSR (0.64) HTR1AHTR1DHTR1BGPR84CTSV
SCHEMBL532789 0.75 HTR1A (0.55) HTR1AHTR1DHTR1BGABRA1GABRB2
SCHEMBL2421287 0.74 GPR84 (0.54) GPR84
SCHEMBL12100781 0.74 HTR1A (0.57) HTR1AHTR1DHTR1BCTSVCTSL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009103007-A2 STEROID HORMONE RECEPTOR MODULATOR COMPOUNDS AND METHODS LIGAND PHARMACEUTICALS INCORPORATED (US) 2009-08-20 WO disclosed