SCHEMBL4510544

SCHEMBL4510544

[c]1nc(-c2cnc3ccccc3n2)c2ccccc2n1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 6/20 0.45
ADORA1 P30542 3/20 0.45
ADORA2A P29274 2/20 0.45
NPC1 O15118 7/20 0.44
RAB9A P51151 5/20 0.44
SMN1; SMN2 Q16637 3/20 0.44
BCHE P06276 1/20 0.44
KDM4E B2RXH2 4/20 0.43
GPR3 P46089 1/20 0.43
ALDH1A1 P00352 3/20 0.42
MAPK10 P53779 2/20 0.42
HPGD P15428 2/20 0.42
GAA P10253 1/20 0.42
CASP1 P29466 1/20 0.42
CASP7 P55210 1/20 0.42
HSD17B10 Q99714 1/20 0.42
CYP1A2 P05177 1/20 0.40
MAPT P10636 3/20 0.39
PDE10A Q9Y233 1/20 0.38
MEN1 O00255 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4512439 0.80 NPC1 (0.50) ADORA3ADORA1ADORA2ANPC1RAB9A
SCHEMBL14941820 0.78 RAB9A (0.43) NPC1RAB9ASMN1; SMN2KDM4EALDH1A1
SCHEMBL21023293 0.76 ADORA2A (0.55) ADORA3ADORA1ADORA2ANPC1RAB9A
SCHEMBL28395491 0.76 NPC1 (0.57) ADORA3ADORA1ADORA2ANPC1RAB9A
SCHEMBL1558294 0.75 BCHE (0.36) ADORA3ADORA1ADORA2ANPC1RAB9A
SCHEMBL9265475 0.74 KDM4E (0.36) ADORA3ADORA1ADORA2ANPC1RAB9A
SCHEMBL29614829 0.73 NPC1 (0.63) ADORA3ADORA1ADORA2ANPC1RAB9A
SCHEMBL29942654 0.73 NPC1 (0.63) ADORA3ADORA1ADORA2ANPC1RAB9A
SCHEMBL29966674 0.73 NPC1 (0.63) ADORA3ADORA1ADORA2ANPC1RAB9A
SCHEMBL3076524 0.73 NPC1 (0.63) ADORA3ADORA1ADORA2ANPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117529202-A Organometallic compound, light-emitting device, electronic apparatus, and electronic device 三星显示有限公司 2024-02-06 CN disclosed
CN-115701262-A Organic light emitting device 三星电子株式会社 2023-02-07 CN disclosed
US-9255091-B2 Benzothiazole-based pyridinium compounds THE UNIVERSITY OF MONTANA (US) 2016-02-09 US disclosed
EP-2948129-A1 THERAPEUTIC COMPOUNDS Wintermute Biomedical LLC (US) 2015-12-02 EP disclosed
US-20150259336-A1 Benzothiazole-based Pyridinium Compounds for the Treatment of Neurodegenerative Diseases or Nerve Agent Exposure THE UNIVERSITY OF MONTANA (US) 2015-09-17 US disclosed
WO-2014117056-A1 THERAPEUTIC COMPOUNDS WINTERMUTE BIOMEDICAL, LLC (US) 2014-07-31 WO disclosed
US-20090023728-A1 1,2,3,4-Tetrahydroisoquinoline Derivatives, Preparations Thereof and Uses Thereof ASTRAZENECA AB (SE) 2009-01-22 US disclosed
US-6335345-B1 NEUROPEPTIDE Y RECEPTOR ANTAGONISTS; OBESITY AND BULIMIA TREATMENT; CENTRAL NERVOUS SYSTEM, PSYCHOLOGICAL, METABOLIC AND EATING DISORDERS; ANTIDIABETIC AGENTS BANYU PHARMACEUTICAL CO., LTD. (JP) 2002-01-01 US disclosed
US-6147051-A ANTIISCHEMIC AGENT TAKEDA CHEMICAL INDUSTRIES LTD. (JP) 2000-11-14 US disclosed
EP-0626174-A2 Methods and compositions for the prophylactic and/or therapeutic treatment of organ hypofunction TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1994-11-30 EP disclosed
US-4902800-A USED AS ANTIINFLAMMATORY AGENTS AND IN TREATMENT OF DISEASE STATES INVOLVING ENZYMATIC TISSUE DESTRUCTION AMERICAN HOME PRODUCTS CORPORATION (US) 1990-02-20 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20150259336-A1 Benzothiazole-based Pyridinium Compounds for the Treatment of Neurodegenerative Diseases or Nerve Agent Exposure BCHE, ACHE, BACE1 ADORA3 1875/4885ADORA1 1327/4885ADORA2A 2442/4885
US-20090023728-A1 1,2,3,4-Tetrahydroisoquinoline Derivatives, Preparations Thereof and Uses Thereof OPRD1, QDPR, RECQL ADORA3 381/4885ADORA1 537/4885ADORA2A 836/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.