SCHEMBL4511545

SCHEMBL4511545

COC(=O)C1CCc2nnc(-c3ccccc3)n21

nearest known ligand 0.46

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.45
CYP3A4 P08684 3/20 0.42
KDM4E B2RXH2 2/20 0.42
ALDH1A1 P00352 2/20 0.42
XDH P47989 1/20 0.40
ADRB2 P07550 1/20 0.40
SLC6A4 P31645 2/20 0.39
GAA P10253 2/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
HPGD P15428 1/20 0.38
MAPT P10636 1/20 0.38
SLC6A2 P23975 1/20 0.38
MMP2 P08253 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13628885 0.92 HPGD (0.43) KMT2ACYP3A4KDM4EALDH1A1XDH
SCHEMBL4515035 0.79 FKBP1A (0.44) KMT2ACYP3A4KDM4EALDH1A1L3MBTL1
SCHEMBL23657877 0.70 NPC1 (0.53) KMT2AKDM4EALDH1A1HPGDMAPT
SCHEMBL10189678 0.69 ADRB3 (0.41) KMT2AKDM4EALDH1A1MMP2
SCHEMBL11964111 0.69 ADRB3 (0.41) KMT2AKDM4EALDH1A1MMP2
SCHEMBL1199646 0.68 KMT2A (0.44) KMT2AALDH1A1SLC6A4MMP2
SCHEMBL4507031 0.68 SIGMAR1 (0.36) KMT2ACYP3A4ALDH1A1SLC6A4HPGD
SCHEMBL950990 0.68 KMT2A (0.45) KMT2AKDM4EALDH1A1HPGDMAPT
SCHEMBL23657646 0.67 CNR2 (0.40) KMT2ACYP3A4KDM4EALDH1A1SLC6A4
SCHEMBL27070540 0.66 CYP1A2 (0.40) KMT2ASLC6A4SLC6A2MMP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7618983-B2 Bicyclic triazole α4 integrin inhibitors JANSSEN PHARMACEUTICA, N.V. (BE) 2009-11-17 US disclosed
US-20060128748-A1 Bicyclic triazole alpha4 integrin inhibitors JANSSEN PHARMACEUTICA, N.V. (BE) 2006-06-15 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060128748-A1 Bicyclic triazole alpha4 integrin inhibitors ITGA4, ITGB4, ITGB5 KMT2A 2094/4885CYP3A4 299/4885KDM4E 839/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.