SCHEMBL452453

SCHEMBL452453

O=Cc1cnc2sc(Br)nn12

nearest known ligand 0.33

Predicted protein targets (top 1)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15013254 0.80 RAB9A (0.43) ALDH1A1
SCHEMBL2253505 0.76 LMNA (0.33) ALDH1A1
SCHEMBL15349467 0.73 RAB9A (0.30)
SCHEMBL23292148 0.71 RAB9A (0.30)
SCHEMBL452296 0.71 CHEK1 (0.32)
SCHEMBL2253715 0.68 TNF (0.31)
SCHEMBL7329300 0.62 DCTPP1 (0.39)
SCHEMBL2257307 0.62 ALDH1A1 (0.34) ALDH1A1
SCHEMBL7331691 0.60 CHEK1 (0.49) ALDH1A1
SCHEMBL452454 0.60 F2RL3 (0.40)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011121317-A9 IMIDAZOTHIADIAZOLES FOR USE AS KINASE INHIBITORS CENTRO NACIONAL DE INVESTIGACIONES ONCOLOGICAS (CNIO) (ES) 2012-03-15 WO disclosed
WO-2011121317-A1 IMIDAZO [2,1-B] [1,3,4] THIADIAZOLES AS PROTEIN OR LIPID KINASE INHIBITORS CENTRO NACIONAL DE INVESTIGACIONES ONCOLOGICAS (CNIO) (ES) 2011-10-06 WO disclosed