SCHEMBL4526732

SCHEMBL4526732

CCC[C@H]1CC1(C(=O)OC)C(=O)OC

nearest known ligand 0.36

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.35
CYP3A4 P08684 3/20 0.33
TSHR P16473 3/20 0.33
CYP4F2 P78329 1/20 0.33
CYP4A11 Q02928 1/20 0.33
NPSR1 Q6W5P4 2/20 0.31
LMNA P02545 2/20 0.31
TP53 P04637 2/20 0.31
MAPK1 P28482 1/20 0.31
HTT P42858 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30
L3MBTL1 Q9Y468 1/20 0.30
ALDH1A1 P00352 1/20 0.30
HPGD P15428 1/20 0.30
HSD17B10 Q99714 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9416811 1.00 MAPT (0.35) MAPTCYP3A4TSHRCYP4F2CYP4A11
SCHEMBL9416740 0.91 MAPT (0.35) MAPTCYP3A4TSHRCYP4F2CYP4A11
SCHEMBL4526740 0.91 MAPT (0.35) MAPTCYP3A4TSHRCYP4F2CYP4A11
SCHEMBL30707215 0.83 MAPT (0.36) MAPTCYP4F2CYP4A11NPSR1L3MBTL1
SCHEMBL11783192 0.81 PTPN1 (0.35) MAPTCYP4F2CYP4A11NPSR1ALDH1A1
SCHEMBL14035534 0.80 MAPT (0.34) MAPTCYP4F2CYP4A11HTTALDH1A1
SCHEMBL15483730 0.78 CYP3A4 (0.34) MAPTCYP3A4TSHRNPSR1LMNA
SCHEMBL13757812 0.77 GRM2 (0.36) MAPTCYP3A4TSHRNPSR1LMNA
SCHEMBL3369422 0.77 GRM2 (0.36) MAPTCYP3A4TSHRNPSR1LMNA
SCHEMBL4507473 0.77 GRM2 (0.33)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1993998-B1 3-CARBOXY- 2-OXO-1 -PYRROLIDINE DERIVATIVES AND THEIR USES UCB PHARMA SA (BE) 2013-08-21 EP disclosed
EP-1993998-B1 3-CARBOXY- 2-OXO-1 -PYRROLIDINE DERIVATIVES AND THEIR USES UCB PHARMA SA (BE) 2013-08-21 EP disclosed
US-8076493-B2 3-carboxy-2-oxo-1-pyrrolidine derivatives and their uses UCB PHARMA, S.A. (BE) 2011-12-13 US disclosed
US-8076493-B2 3-carboxy-2-oxo-1-pyrrolidine derivatives and their uses UCB PHARMA, S.A. (BE) 2011-12-13 US disclosed
US-8076493-B2 3-carboxy-2-oxo-1-pyrrolidine derivatives and their uses UCB PHARMA, S.A. (BE) 2011-12-13 US disclosed
US-20090012313-A1 3-Carboxy-2-Oxo-1-Pyrrolidine Derivatives and Their Uses UCB PHARMA, S.A. (BE) 2009-01-08 US disclosed
US-20090012313-A1 3-Carboxy-2-Oxo-1-Pyrrolidine Derivatives and Their Uses UCB PHARMA, S.A. (BE) 2009-01-08 US disclosed
US-20090012313-A1 3-Carboxy-2-Oxo-1-Pyrrolidine Derivatives and Their Uses UCB PHARMA, S.A. (BE) 2009-01-08 US disclosed
EP-1993998-A1 3-CARBOXY- 2-OXO-1 -PYRROLIDINE DERIVATIVES AND THEIR USES UCB Pharma, S.A. (BE) 2008-11-26 EP disclosed
WO-2007065634-A1 3-CARBOXY- 2-OXO-1 -PYRROLIDINE DERIVATIVES AND THEIR USES UCB PHARMA, S.A. (BE) 2007-06-14 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090012313-A1 3-Carboxy-2-Oxo-1-Pyrrolidine Derivatives and Their Uses ALDH18A1, PYCR1, OPRD1 MAPT 3528/4885CYP3A4 24/4885TSHR 4398/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.