SCHEMBL4534819

SCHEMBL4534819

CC(=O)Nc1ccc(S(=O)(=O)N2CCCCC2CNC(=O)C23CC4CC(CC(C4)C2)C3)cc1

nearest known ligand 0.54

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.54
POLB P06746 1/20 0.54
MEN1 O00255 2/20 0.50
KMT2A Q03164 2/20 0.50
RAB9A P51151 1/20 0.50
PAX8 Q06710 1/20 0.50
ADRB2 P07550 1/20 0.48
TSHR P16473 1/20 0.48
NAMPT P43490 2/20 0.47
LMNA P02545 2/20 0.47
MAPT P10636 1/20 0.47
SMN1; SMN2 Q16637 2/20 0.46
NPC1 O15118 2/20 0.45
AKR1C3 P42330 1/20 0.45
CA12 O43570 1/20 0.45
CA9 Q16790 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4535257 0.88 RAB9A (0.53) ALDH1A1RAB9APAX8TSHR
SCHEMBL4539052 0.86 ALDH1A1 (0.47) ALDH1A1RAB9APAX8TSHR
SCHEMBL4536842 0.86 RAB9A (0.50) ALDH1A1RAB9ATSHRMAPTSMN1; SMN2
SCHEMBL4535933 0.86 PSEN1 (0.56) ALDH1A1PAX8TSHRLMNA
SCHEMBL4537565 0.86 RAB9A (0.51) ALDH1A1RAB9ANPC1
SCHEMBL4541154 0.85 RAB9A (0.56) RAB9APAX8
SCHEMBL8069510 0.84 BRD4 (0.53) ALDH1A1
SCHEMBL4538787 0.83 PSEN1 (0.51) POLBPAX8TSHRLMNA
SCHEMBL4535339 0.83 ATM (0.47) RAB9APAX8LMNASMN1; SMN2
SCHEMBL4542333 0.83 PSEN1 (0.51) POLBPAX8TSHRLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009070497-A1 SEH AND 11 β-HSD1 INHIBITORS AND THEIR USE SMITHKLINE BEECHAM CORPORATION (US) 2009-06-04 WO claimed
WO-2009070497-A1 SEH AND 11 β-HSD1 INHIBITORS AND THEIR USE SMITHKLINE BEECHAM CORPORATION (US) 2009-06-04 WO disclosed