SCHEMBL4535231

SCHEMBL4535231

Cc1cccc(S(=O)(=O)N2CCC[C@@H]2CC(=O)NC23CC4CC(CC(C4)C2)C3)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR7 P34969 4/20 0.52
HTR1B P28222 3/20 0.52
DRD3 P35462 3/20 0.52
HTR1A P08908 2/20 0.52
DRD2 P14416 2/20 0.52
HTR1D P28221 2/20 0.52
EPHX2 P34913 3/20 0.44
USP2 O75604 1/20 0.44
LMNA P02545 1/20 0.44
SMN1; SMN2 Q16637 2/20 0.43
RAB9A P51151 2/20 0.43
NPC1 O15118 1/20 0.43
KMT2A Q03164 1/20 0.43
EPHX1 P07099 1/20 0.43
CYP2D6 P10635 2/20 0.42
HTR5A P47898 2/20 0.42
CYP3A4 P08684 1/20 0.42
CYP1A2 P05177 1/20 0.42
HTR2B P41595 1/20 0.42
HTR6 P50406 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4542494 1.00 HTR7 (0.52) HTR7HTR1BDRD3HTR1ADRD2
SCHEMBL4537661 0.97 HTR1A (0.48) HTR7HTR1BDRD3HTR1ADRD2
SCHEMBL4541345 0.89 POLB (0.44) HTR7HTR1BDRD3HTR1ADRD2
SCHEMBL4536998 0.89 BDKRB1 (0.49) HTR7HTR1BDRD3HTR1ADRD2
SCHEMBL4541024 0.88 RAB9A (0.48) EPHX2LMNARAB9AEPHX1BDKRB1
SCHEMBL4542819 0.88 RAB9A (0.54) EPHX2SMN1; SMN2RAB9ANPC1KMT2A
SCHEMBL4535169 0.88 HTR7 (0.54) HTR7EPHX2USP2LMNARAB9A
SCHEMBL8058321 0.88 HTR7 (0.46) HTR7HTR1BDRD3HTR1ADRD2
SCHEMBL8064947 0.87 HTR1A (0.50) HTR7HTR1BDRD3HTR1ADRD2
SCHEMBL4537195 0.87 HTR1A (0.50) HTR7HTR1BDRD3HTR1ADRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009070497-A1 SEH AND 11 β-HSD1 INHIBITORS AND THEIR USE SMITHKLINE BEECHAM CORPORATION (US) 2009-06-04 WO claimed
WO-2009070497-A1 SEH AND 11 β-HSD1 INHIBITORS AND THEIR USE SMITHKLINE BEECHAM CORPORATION (US) 2009-06-04 WO disclosed