SCHEMBL4535499

SCHEMBL4535499

O=C(NCC1CCN(S(=O)(=O)c2ccc(F)cc2)CC1)C12CC3CC(CC(C3)C1)C2

nearest known ligand 0.56

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.56
POLB P06746 2/20 0.50
TP53 P04637 1/20 0.50
PKM P14618 2/20 0.47
L3MBTL1 Q9Y468 2/20 0.47
KMT2A Q03164 2/20 0.47
USP5 P45974 1/20 0.47
NAMPT P43490 1/20 0.47
ENPP3 O14638 1/20 0.47
CA12 O43570 1/20 0.47
ENPP1 P22413 1/20 0.47
ENPP2 Q13822 1/20 0.47
CA9 Q16790 1/20 0.47
EPHX2 P34913 1/20 0.47
KDM4E B2RXH2 2/20 0.46
GAA P10253 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4541335 0.94 CYP3A4 (0.51) ALDH1A1POLBTP53PKMKMT2A
SCHEMBL8066749 0.94 CYP3A4 (0.51) ALDH1A1POLBTP53PKMKMT2A
SCHEMBL4541776 0.89 LMNA (0.55) ALDH1A1POLBL3MBTL1KMT2AUSP5
SCHEMBL4541037 0.89 ALDH1A1 (0.61) ALDH1A1PKML3MBTL1KMT2AEPHX2
SCHEMBL4535774 0.89 CYP3A4 (0.59) ALDH1A1TP53KMT2ANAMPT
SCHEMBL4542839 0.86 PKM (0.56) ALDH1A1PKMKMT2AUSP5EPHX2
SCHEMBL4534658 0.85 CYP3A4 (0.49) ALDH1A1POLBTP53PKMKMT2A
SCHEMBL8064991 0.83 ALDH1A1 (0.49) ALDH1A1POLBL3MBTL1KMT2ACA12
SCHEMBL8061563 0.83 LMNA (0.51) ALDH1A1POLBKMT2AEPHX2KDM4E
SCHEMBL4532816 0.83 TP53 (0.48) ALDH1A1POLBTP53PKMKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009070497-A1 SEH AND 11 β-HSD1 INHIBITORS AND THEIR USE SMITHKLINE BEECHAM CORPORATION (US) 2009-06-04 WO disclosed
WO-2009070497-A1 SEH AND 11 β-HSD1 INHIBITORS AND THEIR USE SMITHKLINE BEECHAM CORPORATION (US) 2009-06-04 WO disclosed