SCHEMBL8066749

SCHEMBL8066749

O=C(NCC1CCN(S(=O)(=O)c2ccc(F)cc2)C1)C12CC3C[C@H](C1)C[C@@H](C3)C2

nearest known ligand 0.51

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.51
CYP2C19 P33261 1/20 0.51
ALDH1A1 P00352 3/20 0.49
TP53 P04637 2/20 0.48
POLB P06746 1/20 0.48
MAPT P10636 1/20 0.46
NAMPT P43490 1/20 0.45
ENPP3 O14638 1/20 0.45
CA12 O43570 1/20 0.45
ENPP1 P22413 1/20 0.45
ENPP2 Q13822 1/20 0.45
CA9 Q16790 1/20 0.45
KMT2A Q03164 4/20 0.44
PKM P14618 1/20 0.44
P2RX7 Q99572 1/20 0.44
MEN1 O00255 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
USP5 P45974 1/20 0.43
SLC13A5 Q86YT5 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4541335 1.00 CYP3A4 (0.51) CYP3A4CYP2C19ALDH1A1TP53POLB
SCHEMBL4535774 0.95 CYP3A4 (0.59) CYP3A4CYP2C19ALDH1A1TP53MAPT
SCHEMBL4535499 0.94 ALDH1A1 (0.56) ALDH1A1TP53POLBNAMPTENPP3
SCHEMBL8064991 0.90 ALDH1A1 (0.49) ALDH1A1POLBCA12CA9KMT2A
SCHEMBL4534658 0.90 CYP3A4 (0.49) CYP3A4CYP2C19ALDH1A1TP53POLB
SCHEMBL4535269 0.89 LMNA (0.51) ALDH1A1POLBKMT2AMEN1SMN1; SMN2
SCHEMBL4532816 0.89 TP53 (0.48) ALDH1A1TP53POLBKMT2APKM
SCHEMBL4531159 0.89 ALDH1A1 (0.51) ALDH1A1POLBCA12CA9KMT2A
SCHEMBL8061563 0.89 LMNA (0.51) ALDH1A1POLBKMT2AMEN1SMN1; SMN2
SCHEMBL4542831 0.89 ALDH1A1 (0.53) ALDH1A1ENPP3ENPP1ENPP2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009070497-A1 SEH AND 11 β-HSD1 INHIBITORS AND THEIR USE SMITHKLINE BEECHAM CORPORATION (US) 2009-06-04 WO disclosed