SCHEMBL4537013

SCHEMBL4537013

COc1ccccc1S(=O)(=O)N1CCC(CNC(=O)N[C]2CCCCCCC2)C1.[CH2].[CH2]

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 11/20 0.44
L3MBTL1 Q9Y468 2/20 0.44
MAPT P10636 5/20 0.43
KDM4E B2RXH2 3/20 0.43
MCL1 Q07820 3/20 0.43
HPGD P15428 2/20 0.43
TDP1 Q9NUW8 2/20 0.43
KMT2A Q03164 3/20 0.43
TSHR P16473 2/20 0.43
HTT P42858 2/20 0.43
MEN1 O00255 2/20 0.43
MAPK1 P28482 1/20 0.43
LMNA P02545 3/20 0.42
ALOX15 P16050 2/20 0.42
USP2 O75604 1/20 0.42
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4539565 0.87 EPHX2 (0.48) ALDH1A1L3MBTL1MAPTKDM4EMCL1
SCHEMBL4537189 0.85 FAAH (0.49) ALDH1A1L3MBTL1
SCHEMBL4537541 0.85 ALDH1A1 (0.52) ALDH1A1L3MBTL1KMT2AMEN1MAPK1
SCHEMBL4542230 0.85 CYP19A1 (0.54) ALDH1A1L3MBTL1MAPTKDM4EMCL1
SCHEMBL4535742 0.83 NPC1 (0.52) ALDH1A1L3MBTL1MAPTKDM4EMCL1
SCHEMBL4539885 0.82 FAAH (0.45) ALDH1A1L3MBTL1POLB
SCHEMBL4539993 0.81 ALDH1A1 (0.51) ALDH1A1L3MBTL1MAPTKDM4EMCL1
SCHEMBL4533514 0.81 ALDH1A1 (0.53) ALDH1A1L3MBTL1KMT2AMEN1BRD4
SCHEMBL4535453 0.80 ALDH1A1 (0.56) ALDH1A1L3MBTL1MAPTKDM4EKMT2A
SCHEMBL4537967 0.79 ALDH1A1 (0.50) ALDH1A1L3MBTL1KMT2ATSHRMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009070497-A1 SEH AND 11 β-HSD1 INHIBITORS AND THEIR USE SMITHKLINE BEECHAM CORPORATION (US) 2009-06-04 WO claimed
WO-2009070497-A1 SEH AND 11 β-HSD1 INHIBITORS AND THEIR USE SMITHKLINE BEECHAM CORPORATION (US) 2009-06-04 WO disclosed