SCHEMBL4538265

SCHEMBL4538265

CC(C)[N+](C)(CCC(C(N)=O)(c1ccccc1)c1ccccc1)C(C)CI

nearest known ligand 0.80

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM3 P20309 8/20 0.80
CHRM2 P08172 5/20 0.80
KCNH2 Q12809 3/20 0.80
LMNA P02545 1/20 0.80
CYP2D6 P10635 1/20 0.80
CHRM1 P11229 1/20 0.80
KDM4E B2RXH2 1/20 0.78
CTDSP1 Q9GZU7 1/20 0.78
OPRK1 P41145 2/20 0.40
SLC22A2 O15244 1/20 0.40
SLC22A1 O15245 1/20 0.40
PGR P06401 1/20 0.40
THRB P10828 1/20 0.40
ADRB3 P13945 1/20 0.40
BLM P54132 1/20 0.40
PMP22 Q01453 1/20 0.40
PDE3A Q14432 1/20 0.40
SLC47A1 Q96FL8 1/20 0.40
CYP3A4 P08684 1/20 0.40
ALOX15 P16050 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Isopropamide SCHEMBL100256 0.89 CHRM3 (1.00) CHRM3CHRM2KCNH2LMNACYP2D6
Isopropamide SCHEMBL3082703 0.88 CHRM3 (0.97) CHRM3CHRM2KCNH2LMNACYP2D6
Isopropamide SCHEMBL100255 0.88 KDM4E (1.00) CHRM3CHRM2KCNH2LMNACYP2D6
Isopropamide SCHEMBL14672609 0.87 CHRM3 (0.94) CHRM3CHRM2KCNH2LMNACYP2D6
Isopropamide SCHEMBL7796559 0.82 CHRM3 (0.85) CHRM3CHRM2KCNH2LMNACYP2D6
Isopropamide SCHEMBL17923572 0.78 KDM4E (0.79) CHRM3CHRM2KCNH2LMNACYP2D6
Ambutonium SCHEMBL11946672 0.74 CHRM3 (0.67) CHRM3CHRM2KCNH2LMNACYP2D6
Ambutonium SCHEMBL249674 0.72 CHRM3 (0.65) CHRM3CHRM2KCNH2LMNACYP2D6
SCHEMBL6834396 0.71 CHRM3 (0.56) CHRM3CHRM2KCNH2LMNACYP2D6
SCHEMBL25341236 0.71 CHRM3 (0.63) CHRM3CHRM2KCNH2LMNACYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115916305-A Multi-carrier medicament dispenser 陆品公司 2023-04-04 CN disclosed
CN-108033921-B 3, 5-diamino-6-chloro-N- (N- (4- (4- (2- (hexyl (2,3,4,5, 6-pentahydroxyhexyl) amino) ethoxy) phenyl) butyl) carbamimidoyl) pyrazine-2-carboxamide 帕里昂科学公司 2021-07-20 CN disclosed
JP-2009197011-A ANTIRHEUMIC AGENT DAIICHI SANKYO HEALTHCARE CO LTD 2009-09-03 JP disclosed