SCHEMBL4540052

SCHEMBL4540052

Cc1ccc(S(=O)(=O)OCCc2c(S(=O)(=O)c3ccc(C)cc3)[nH]c3cc(Br)ccc23)cc1

nearest known ligand 0.37

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
GPR17 Q13304 1/20 0.37
MCL1 Q07820 2/20 0.37
CHRNB2 P17787 4/20 0.34
CHRNA7 P36544 4/20 0.34
CHRNA4 P43681 4/20 0.34
KMT2A Q03164 2/20 0.34
MEN1 O00255 1/20 0.34
LMNA P02545 1/20 0.34
PKM P14618 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
CA12 O43570 2/20 0.34
CA1 P00915 2/20 0.34
CA2 P00918 1/20 0.34
CA9 Q16790 1/20 0.33
MAPT P10636 2/20 0.32
HTR6 P50406 1/20 0.32
TP53 P04637 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
TDP1 Q9NUW8 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4543731 0.87 POLB (0.40) GPR17MCL1
SCHEMBL4231056 0.84 EGFR (0.46) MCL1HTR6SMN1; SMN2
SCHEMBL4233057 0.84 GPR17 (0.38) GPR17MCL1CHRNB2CHRNA7CHRNA4
SCHEMBL4542962 0.80 POLB (0.45) MCL1KMT2AMEN1MAPTHTR6
SCHEMBL4225100 0.80 MAPT (0.40) KMT2AMEN1NPSR1CA12CA1
SCHEMBL4233003 0.80 MAPT (0.50) KMT2AMEN1LMNAMAPTHTR6
SCHEMBL4223972 0.78 GPR17 (0.37) GPR17MCL1KMT2ALMNACA12
SCHEMBL4219372 0.75 LMNA (0.41) KMT2AMEN1LMNAPKMNPSR1
SCHEMBL828951 0.73 EGFR (0.47) KMT2AMEN1CA12CA1CA2
SCHEMBL24598179 0.71 THRB (0.42) KMT2AMEN1LMNAPKMNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009006089-A2 A2 ADENOSINE RECEPTOR AGONISTS GOVERNMENT OF THE UNITED STATES OF AMERICA, REPRESENTED BY THE SECRETARY, DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 2009-01-08 WO disclosed