SCHEMBL4543170

SCHEMBL4543170

O=S(=O)(OCCCOCc1ccccc1)C(F)(F)F

nearest known ligand 0.46

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CA2 P00918 3/20 0.46
CA1 P00915 2/20 0.44
TSHR P16473 1/20 0.44
CA9 Q16790 1/20 0.43
TDP1 Q9NUW8 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
MGLL Q99685 1/20 0.40
CES1 P23141 1/20 0.40
HRH4 Q9H3N8 1/20 0.39
HRH3 Q9Y5N1 1/20 0.39
PTPN2 P17706 1/20 0.39
PTPN1 P18031 1/20 0.39
PTPN6 P29350 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21068846 0.98 CA2 (0.45) CA2CA1TSHRCA9TDP1
SCHEMBL9107341 0.90 CA2 (0.49) CA2CA1TSHRCA9MGLL
SCHEMBL29287385 0.83 TSHR (0.50) CA2CA1TSHRCA9TDP1
SCHEMBL4625553 0.81 CA2 (0.55) CA2CA1CA9CES1
SCHEMBL777315 0.81 CA2 (0.66) CA2CA1TSHRCA9MGLL
SCHEMBL7399184 0.81 TSHR (0.44) CA2CA1TSHRCA9TDP1
SCHEMBL30123980 0.80 CA2 (0.43) CA2CA1TSHRCA9MGLL
SCHEMBL2076982 0.80 ALDH1A1 (0.47) CA2CA1TSHRCA9TDP1
SCHEMBL8007555 0.80 CA2 (0.54) CA2CA1CA9MGLLCES1
Ammonia Solution, Strong SCHEMBL28512991 0.79 CA2 (0.64) CA2CA1TSHRCA9MGLL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012062229-A1 A METHOD OF MANUFACTURING (-)-L-(3-HYDROXYPROPYL)-5-[(2R)-2-({2,2,2-TRIFLUOROETHOXY)- PHENOXYETHYL}AMINO)PROPYL]-2,3-DIHYDRO-LH-INDOLE-7-CARBOXAMIDE ZENTIVA, K.S. (CZ) 2012-05-18 WO disclosed