SCHEMBL4553008

SCHEMBL4553008

CCCc1ccc(I)nn1

nearest known ligand 0.39

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 2/20 0.33
KDM4E B2RXH2 1/20 0.32
LMNA P02545 1/20 0.32
CYP3A4 P08684 1/20 0.32
TSHR P16473 1/20 0.32
NOS3 P29474 1/20 0.31
NOS1 P29475 1/20 0.31
NOS2 P35228 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19009140 0.78 CYP19A1 (0.36) CYP19A1KDM4ELMNACYP3A4TSHR
SCHEMBL19009143 0.76 KCNH2 (0.45) CYP19A1NOS2
SCHEMBL21690815 0.76 CYP19A1 (0.33) CYP19A1KDM4ELMNACYP3A4TSHR
SCHEMBL17858892 0.74 NOS2 (0.36) CYP19A1KDM4ELMNACYP3A4TSHR
SCHEMBL10841047 0.73 CYP19A1 (0.33) CYP19A1KDM4ELMNACYP3A4TSHR
SCHEMBL12678552 0.73 NOS2 (0.44) CYP19A1KDM4ELMNACYP3A4TSHR
SCHEMBL3182612 0.73 ALDH1A1 (0.48) CYP19A1KDM4ELMNACYP3A4TSHR
SCHEMBL18647537 0.71 NOS3 (0.39) CYP19A1KDM4ELMNACYP3A4TSHR
SCHEMBL255651 0.71
SCHEMBL25913119 0.69 CYP19A1 (0.31) CYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2121600-A2 SUBSTITUTED ARYLSULPHONYLGLYCINES, THE PREPARATION THEREOF AND THE USE THEREOF AS PHARMACEUTICAL COMPOSITIONS Boehringer Ingelheim International GmbH (DE) 2009-11-25 EP disclosed
WO-2008099000-A2 SUBSTITUTED ARYLSULPHONYLGLYCINES, THE PREPARATION THEREOF AND THE USE THEREOF AS PHARMACEUTICAL COMPOSITIONS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2008-08-21 WO disclosed