SCHEMBL4553444

SCHEMBL4553444

Cc1nn(C)c(-n2ccc3cc(Cl)ccc32)c1CCS(=O)(=O)NC(=O)OCc1ccccc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.44
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
PTGER1 P34995 1/20 0.37
PTGDR2 Q9Y5Y4 3/20 0.37
CYP1A2 P05177 2/20 0.36
CYP2C19 P33261 2/20 0.36
GALR3 O60755 1/20 0.36
CYP3A4 P08684 1/20 0.36
HTT P42858 1/20 0.36
BRD4 O60885 1/20 0.36
BRD2 P25440 1/20 0.36
BRD3 Q15059 1/20 0.36
MCL1 Q07820 1/20 0.36
PLA2G4A P47712 5/20 0.35
PPARG P37231 1/20 0.35
CA12 O43570 1/20 0.35
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35
CA9 Q16790 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4555122 0.91 MAPK8 (0.37) SMN1; SMN2CYP1A2CYP2C19GALR3CYP3A4
SCHEMBL4570493 0.88 PHGDH (0.36) MEN1KMT2APTGDR2MCL1PLA2G4A
SCHEMBL4553883 0.87 SMN1; SMN2 (0.33) SMN1; SMN2MEN1KMT2ACYP1A2CYP2C19
SCHEMBL4554740 0.87 AGTR2 (0.37) MCL1PLA2G4APPARG
SCHEMBL4554652 0.86 GABRA1 (0.36) SMN1; SMN2CYP1A2CYP2C19GALR3CYP3A4
SCHEMBL4554828 0.84 AGTR2 (0.38) SMN1; SMN2CYP1A2CYP2C19GALR3CYP3A4
SCHEMBL963395 0.83 KMT2A (0.37) SMN1; SMN2MEN1KMT2APTGDR2PLA2G4A
SCHEMBL4554438 0.82 MAPK8 (0.35) SMN1; SMN2CYP1A2CYP2C19GALR3CYP3A4
SCHEMBL4554288 0.81 TP53 (0.38) SMN1; SMN2MEN1KMT2ACYP1A2CYP2C19
SCHEMBL5115435 0.81 KMO (0.38) SMN1; SMN2KMT2APTGDR2CYP1A2CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2118066-A1 FUSED RING COMPOUNDS AS PARTIAL AGONISTS OF PPAR-GAMMA Takeda Pharmaceutical Company Limited (JP) 2009-11-18 EP disclosed
WO-2008099794-A1 FUSED RING COMPOUNDS AS PARTIAL AGONISTS OF PPAR-GAMMA TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2008-08-21 WO disclosed