SCHEMBL4553763

SCHEMBL4553763

CCCCC(CS(=O)(=O)OC(N)=O)c1c(C)nn(C)c1-n1ccc2ccc(Cl)cc21

nearest known ligand 0.31

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ADA P00813 2/20 0.31
KMO O15229 1/20 0.31
NPY5R Q15761 1/20 0.30
CRHR1 P34998 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4554440 0.95 KMO (0.31) KMONPY5R
SCHEMBL4554742 0.94 MAPK8 (0.31) ADANPY5RCRHR1
SCHEMBL4554506 0.86 NPY5R (0.38) KMONPY5R
SCHEMBL4554830 0.85 OXER1 (0.31)
SCHEMBL4555123 0.85 MAPK8 (0.33) NPY5RCRHR1
SCHEMBL4553761 0.82 MAPK8 (0.31) KMOCRHR1
SCHEMBL4553884 0.81 IRAK4 (0.33) NPY5R
SCHEMBL4554653 0.80 NPY5R (0.38) NPY5R
SCHEMBL4553446 0.80 MEN1 (0.40)
SCHEMBL4555092 0.79 POLB (0.34)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2118066-A1 FUSED RING COMPOUNDS AS PARTIAL AGONISTS OF PPAR-GAMMA Takeda Pharmaceutical Company Limited (JP) 2009-11-18 EP disclosed
WO-2008099794-A1 FUSED RING COMPOUNDS AS PARTIAL AGONISTS OF PPAR-GAMMA TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2008-08-21 WO disclosed