SCHEMBL4554830

SCHEMBL4554830

Cc1nn(C)c(-n2ccc3cc(Cl)ccc32)c1C(CCCC(F)(F)F)CS(=O)(=O)OC(N)=O

nearest known ligand 0.31

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
OXER1 Q8TDS5 1/20 0.31
IRAK4 Q9NWZ3 1/20 0.30
PHGDH O43175 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4554742 0.91 MAPK8 (0.31) PHGDH
SCHEMBL4553884 0.91 IRAK4 (0.33) IRAK4PHGDH
SCHEMBL4555123 0.88 MAPK8 (0.33) PHGDH
SCHEMBL4553763 0.85 ADA (0.31)
SCHEMBL4553446 0.84 MEN1 (0.40) PHGDH
SCHEMBL4554653 0.84 NPY5R (0.38) PHGDH
SCHEMBL4554440 0.83 KMO (0.31)
SCHEMBL4554827 0.83 OXER1 (0.31) OXER1IRAK4PHGDH
SCHEMBL4554506 0.78 NPY5R (0.38)
SCHEMBL4553882 0.77 IRAK4 (0.33) IRAK4PHGDH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2118066-A1 FUSED RING COMPOUNDS AS PARTIAL AGONISTS OF PPAR-GAMMA Takeda Pharmaceutical Company Limited (JP) 2009-11-18 EP disclosed
WO-2008099794-A1 FUSED RING COMPOUNDS AS PARTIAL AGONISTS OF PPAR-GAMMA TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2008-08-21 WO disclosed