SCHEMBL4555362

SCHEMBL4555362

NC(=O)c1ccc([C@H]2CC(C3CCNCC3)CCN2C(=O)O)cc1

nearest known ligand 0.43

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
L3MBTL3 Q96JM7 2/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
OPRD1 P41143 1/20 0.39
PARP10 Q53GL7 2/20 0.38
PARP14 Q460N5 1/20 0.38
HRH3 Q9Y5N1 2/20 0.35
GPR119 Q8TDV5 1/20 0.35
CFB P00751 3/20 0.34
CCNC P24863 1/20 0.34
CDK8 P49336 1/20 0.34
SMYD3 Q9H7B4 1/20 0.33
MBTD1 Q05BQ5 1/20 0.33
CYP2C9 P11712 1/20 0.33
ITGB3 P05106 1/20 0.32
ITGA2B P08514 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4554607 0.83 L3MBTL3 (0.38) L3MBTL3L3MBTL1ITGB3ITGA2B
SCHEMBL4555067 0.81 L3MBTL3 (0.38) L3MBTL3L3MBTL1CFBSMYD3ITGB3
SCHEMBL4553619 0.79 LRRK2 (0.38) L3MBTL3L3MBTL1CCNCCDK8
SCHEMBL29213871 0.75 ALDH1A1 (0.49)
SCHEMBL26693343 0.74 PARP14 (0.52) PARP10PARP14HRH3CCNCCDK8
SCHEMBL26693337 0.74 PARP14 (0.52) PARP10PARP14HRH3CCNCCDK8
SCHEMBL4553277 0.74 MAPT (0.35) L3MBTL3L3MBTL1CYP2C9
SCHEMBL26693398 0.73 PARP14 (0.57) PARP10PARP14HRH3CFBCCNC
SCHEMBL4433462 0.73 PKM (0.34) L3MBTL3L3MBTL1CYP2C9
SCHEMBL4555039 0.71 GPR119 (0.48) GPR119

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2121661-A1 BIPIPERIDINYL COMPOUNDS, COMPOSITIONS CONTAINING SUCH COMPOUNDS AND METHODS OF TREATMENT Merck & Co., Inc. (US) 2009-11-25 EP disclosed
WO-2008085316-A1 BIPIPERIDINYL COMPOUNDS, COMPOSITIONS CONTAINING SUCH COMPOUNDS AND METHODS OF TREATMENT MERCK & CO., INC. (US) 2008-07-17 WO disclosed