SCHEMBL4557720

SCHEMBL4557720

NC(=S)N(Cc1cccnc1)/N=C/c1ccc(-c2ccc(F)c(C(F)(F)F)c2)o1

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 3/20 0.38
CYP3A4 P08684 3/20 0.38
KDM4E B2RXH2 2/20 0.37
POLB P06746 2/20 0.37
MAPT P10636 2/20 0.37
HPGD P15428 2/20 0.37
GAA P10253 1/20 0.37
GRIN1 Q05586 2/20 0.37
GRIN2B Q13224 2/20 0.37
VNN1 O95497 1/20 0.36
SIGMAR1 Q99720 1/20 0.35
ALDH1A1 P00352 2/20 0.34
LDHA P00338 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
NAMPT P43490 1/20 0.34
UBE2M P61081 1/20 0.34
DCUN1D1 Q96GG9 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4338180 1.00 CYP2A6 (0.38) CYP2A6CYP3A4KDM4EPOLBMAPT
SCHEMBL4343237 0.86 SIGMAR1 (0.51) CYP2A6CYP3A4KDM4EPOLBMAPT
SCHEMBL4329107 0.84 ALDH1A1 (0.45) CYP2A6CYP3A4KDM4EPOLBMAPT
SCHEMBL4333822 0.83 ALDH1A1 (0.50) CYP2A6CYP3A4KDM4EPOLBMAPT
SCHEMBL4334594 0.83 MAPT (0.46) CYP2A6CYP3A4KDM4EPOLBMAPT
SCHEMBL4338798 0.83 CYP2A6 (0.48) CYP2A6CYP3A4KDM4EPOLBMAPT
SCHEMBL4333786 0.82 SLC9A1 (0.38) CYP2A6CYP3A4POLBMAPTALDH1A1
SCHEMBL4331909 0.81 CYP2A6 (0.43) CYP2A6CYP3A4KDM4EPOLBMAPT
SCHEMBL4329428 0.81 CYP2A6 (0.43) CYP2A6CYP3A4KDM4EPOLBMAPT
SCHEMBL4340661 0.81 CYP2A6 (0.42) CYP2A6CYP3A4KDM4EPOLBMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7521062-B2 Thiosemicarbazones as anti-virals and immunopotentiators NOVARTIS VACCINES & DIAGNOSTICS, INC. (US) 2009-04-21 US disclosed