SCHEMBL4563012

SCHEMBL4563012

CN(C)C(=O)C1CCN(C2CN(C(c3ccccc3)c3ccccc3)C2)CC1.O=C(O)C1CCN(C2CN(C(c3ccccc3)c3ccccc3)C2)CC1

nearest known ligand 0.43

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.43
L3MBTL3 Q96JM7 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
OPRD1 P41143 2/20 0.43
KMT2A Q03164 3/20 0.42
MEN1 O00255 2/20 0.42
POLB P06746 1/20 0.42
CNR1 P21554 1/20 0.41
CNR2 P34972 1/20 0.41
CCR5 P51681 3/20 0.40
SLC6A9 P48067 1/20 0.40
CYP46A1 Q9Y6A2 1/20 0.39
NOTUM Q6P988 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL493703 0.96 ALDH1A1 (0.46) ALDH1A1L3MBTL3L3MBTL1OPRD1KMT2A
SCHEMBL493687 0.90 L3MBTL1 (0.51) ALDH1A1L3MBTL3L3MBTL1OPRD1KMT2A
SCHEMBL4175324 0.80 KMT2A (0.49) ALDH1A1OPRD1KMT2AMEN1POLB
SCHEMBL493492 0.80 TDP1 (0.52) ALDH1A1L3MBTL3L3MBTL1OPRD1KMT2A
SCHEMBL5071337 0.79 CCR5 (0.46) ALDH1A1L3MBTL3L3MBTL1OPRD1KMT2A
SCHEMBL27615098 0.77 L3MBTL3 (0.52) ALDH1A1L3MBTL3L3MBTL1CNR1CNR2
SCHEMBL16822513 0.77 L3MBTL3 (0.51) ALDH1A1L3MBTL3L3MBTL1OPRD1KMT2A
SCHEMBL493765 0.77 ALDH1A1 (0.63) ALDH1A1L3MBTL3L3MBTL1KMT2AMEN1
SCHEMBL17888513 0.76 KDM4E (0.59) ALDH1A1KMT2AMEN1
SCHEMBL2430876 0.76 L3MBTL3 (0.48) ALDH1A1L3MBTL3L3MBTL1OPRD1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2024354-A1 1- [ (4- [BENZOYL (METHYL) AMINO]-3- (PHENYL) BUTYL]AZETIDINE DERIVATIVES FOR THE TREATMENT OF GASTROINTESTINAL DISORDERS 1 Albireo AB (SE) 2009-02-18 EP disclosed
WO-2007136324-A1 1- [ (4- [BENZOYL (METHYL) AMINO] -3- (PHENYL) BUTYL] AZETIDINE DERIVATIVES FOR THE TREATMENT OF GASTROINTESTINAL DISORDERS 1 ALBIREO AB (SE) 2007-11-29 WO disclosed