SCHEMBL2430876

SCHEMBL2430876

O=C(O)OC1CCN(C2CN(C(c3ccccc3)c3ccccc3)C2)CC1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
L3MBTL3 Q96JM7 1/20 0.48
L3MBTL1 Q9Y468 1/20 0.48
ALDH1A1 P00352 2/20 0.45
ACHE P22303 3/20 0.44
BCHE P06276 2/20 0.44
CNR1 P21554 1/20 0.42
CNR2 P34972 1/20 0.42
HRH1 P35367 1/20 0.42
CCR3 P51677 1/20 0.42
KCNH2 Q12809 1/20 0.42
TP53 P04637 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
PKM P14618 1/20 0.41
NFKB1 P19838 1/20 0.41
THPO P40225 1/20 0.41
HIF1A Q16665 1/20 0.41
OPRD1 P41143 1/20 0.41
KMT2A Q03164 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL250850 0.82 ACHE (0.54) ALDH1A1ACHECNR1CNR2KMT2A
SCHEMBL493687 0.82 L3MBTL1 (0.51) L3MBTL3L3MBTL1ALDH1A1CNR1CNR2
SCHEMBL4261834 0.80 L3MBTL3 (0.55) L3MBTL3L3MBTL1ALDH1A1CNR1CNR2
SCHEMBL493492 0.80 TDP1 (0.52) L3MBTL3L3MBTL1ALDH1A1CNR1CNR2
SCHEMBL493703 0.79 ALDH1A1 (0.46) L3MBTL3L3MBTL1ALDH1A1CNR1CNR2
SCHEMBL7467378 0.78 L3MBTL3 (0.57) L3MBTL3L3MBTL1ALDH1A1CNR1CNR2
SCHEMBL16099153 0.77 KMT2A (0.53) L3MBTL3L3MBTL1ALDH1A1CNR1CNR2
SCHEMBL5071336 0.76 L3MBTL3 (0.46) L3MBTL3L3MBTL1ALDH1A1CNR1CNR2
SCHEMBL5071337 0.76 CCR5 (0.46) L3MBTL3L3MBTL1ALDH1A1OPRD1KMT2A
SCHEMBL493765 0.76 ALDH1A1 (0.63) L3MBTL3L3MBTL1ALDH1A1CNR1CNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2024354-B1 1- [ (4- [BENZOYL (METHYL) AMINO]-3- (PHENYL) BUTYL]AZETIDINE DERIVATIVES FOR THE TREATMENT OF GASTROINTESTINAL DISORDERS 1 ALBIREO AB (SE) 2011-09-21 EP claimed