SCHEMBL456348

SCHEMBL456348

O=C(CC1CCCN1)c1nc2ccccc2[nH]1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMYD3 Q9H7B4 1/20 0.47
DAGLA Q9Y4D2 2/20 0.46
SMN1; SMN2 Q16637 4/20 0.45
NPC1 O15118 3/20 0.45
RAB9A P51151 3/20 0.45
FAAH O00519 1/20 0.45
HRH4 Q9H3N8 2/20 0.43
CNR2 P34972 1/20 0.43
CHRNA7 P36544 1/20 0.42
TDP1 Q9NUW8 2/20 0.42
POLB P06746 1/20 0.42
AURKA O14965 1/20 0.42
JAK2 O60674 1/20 0.42
ABL1 P00519 1/20 0.42
NTRK1 P04629 1/20 0.42
LCK P06239 1/20 0.42
FYN P06241 1/20 0.42
CSF1R P07333 1/20 0.42
RET P07949 1/20 0.42
IGF1R P08069 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL416541 0.77 ELANE (0.53) SMYD3SMN1; SMN2NPC1RAB9AFAAH
SCHEMBL454902 0.75 MAOB (0.64) FAAHHRH4
SCHEMBL456347 0.74 FAAH (0.47) SMYD3SMN1; SMN2NPC1RAB9AFAAH
SCHEMBL6670417 0.74 IDO1 (0.55) NPC1RAB9AHRH4POLB
SCHEMBL1255702 0.74 IDO1 (0.55) NPC1RAB9AHRH4POLB
SCHEMBL11343167 0.73 KHK (0.52) SMN1; SMN2TDP1POLB
SCHEMBL1901781 0.71 SMN1; SMN2 (0.61) DAGLASMN1; SMN2NPC1RAB9AHRH4
SCHEMBL29414979 0.71 XDH (0.62) SMYD3DAGLASMN1; SMN2NPC1RAB9A
SCHEMBL30831206 0.71 SMN1; SMN2 (0.61) DAGLASMN1; SMN2NPC1RAB9AHRH4
SCHEMBL6039391 0.71 DAGLA (0.57) DAGLASMN1; SMN2NPC1RAB9AFAAH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2613630-A1 HYDROGEN BOND FORMING FLUORO KETOLIDES FOR TREATING DISEASES Cempra Pharmaceuticals, Inc. (US) 2013-07-17 EP disclosed
WO-2012034058-A1 HYDROGEN BOND FORMING FLUORO KETOLIDES FOR TREATING DISEASES CEMPRA PHARMACEUTICALS, INC. (US) 2012-03-15 WO disclosed