Predicted protein targets (top 20)
| gene | UniProt | supporting neighbours | confidence | |
|---|---|---|---|---|
| ▸ | ELANE | P08246 | 1/20 | 0.53 |
| ▸ | FAAH | O00519 | 1/20 | 0.47 |
| ▸ | AURKA | O14965 | 1/20 | 0.45 |
| ▸ | JAK2 | O60674 | 1/20 | 0.45 |
| ▸ | ABL1 | P00519 | 1/20 | 0.45 |
| ▸ | NTRK1 | P04629 | 1/20 | 0.45 |
| ▸ | LCK | P06239 | 1/20 | 0.45 |
| ▸ | FYN | P06241 | 1/20 | 0.45 |
| ▸ | CSF1R | P07333 | 1/20 | 0.45 |
| ▸ | RET | P07949 | 1/20 | 0.45 |
| ▸ | IGF1R | P08069 | 1/20 | 0.45 |
| ▸ | MET | P08581 | 1/20 | 0.45 |
| ▸ | PDGFRB | P09619 | 1/20 | 0.45 |
| ▸ | PIM1 | P11309 | 1/20 | 0.45 |
| ▸ | FGFR1 | P11362 | 1/20 | 0.45 |
| ▸ | PRKACA | P17612 | 1/20 | 0.45 |
| ▸ | KDR | P35968 | 1/20 | 0.45 |
| ▸ | MAP2K2 | P36507 | 1/20 | 0.45 |
| ▸ | CDK8 | P49336 | 1/20 | 0.45 |
| ▸ | GSK3A | P49840 | 1/20 | 0.45 |
Click a target to see other patent compounds predicted against it — the reverse direction, in place.
Similar compounds — the chemically nearest patent molecules
Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.
| Compound | similarity | top predicted | shared targets | |
|---|---|---|---|---|
| SCHEMBL27573147 | 0.78 | SMN1; SMN2 (0.58) | FAAHAURKAJAK2ABL1NTRK1 | |
| SCHEMBL456348 | 0.77 | SMYD3 (0.47) | FAAHAURKAJAK2ABL1NTRK1 | |
| SCHEMBL456347 | 0.77 | FAAH (0.47) | FAAHAURKAJAK2ABL1NTRK1 | |
| SCHEMBL27553073 | 0.77 | ELANE (0.47) | ELANEFAAHGSK3AGSK3BSMN1; SMN2 | |
| SCHEMBL7469771 | 0.77 | SMN1; SMN2 (0.49) | FAAHAURKAJAK2ABL1NTRK1 | |
| Iodide SCHEMBL7947067 | 0.76 | SMN1; SMN2 (0.48) | FAAHAURKAJAK2ABL1NTRK1 | |
| SCHEMBL1444156 | 0.74 | MAOB (0.52) | ELANECNR2SMN1; SMN2NPC1RAB9A | |
| SCHEMBL28078689 | 0.72 | AURKA (0.51) | FAAHAURKAJAK2ABL1NTRK1 | |
| SCHEMBL250171 | 0.71 | CCND3 (0.70) | FAAHAURKAJAK2ABL1NTRK1 | |
| SCHEMBL741003 | 0.71 | POLB (0.54) | POLB |
Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.
Patent provenance — the patents this molecule appears in, and who filed them
Claimed or disclosed in 175 patents. claimed = in the patent's claims; disclosed = body only.
| Patent | Title | Assignee | Published | Priority | Filing | Country | Status |
|---|---|---|---|---|---|---|---|
| EP-1675474-B9 | PALATABLE DUCTILE CHEWABLE VETERINARY COMPOSITION | NOVARTIS TIERGESUNDHEIT AG (CH) | 2018-12-05 | — | — | EP | claimed |
| US-20170136080-A1 | NOVEL METHOD FOR THE TOPICAL APPLICATION OF VETERINARY AGENTS | Ceva Santé Animale (FR) | 2017-05-18 | — | — | US | claimed |
| EP-3160506-A1 | NOVEL METHOD FOR THE TOPICAL APPLICATION OF VETERINARY AGENTS | Ceva Sante Animale (FR) | 2017-05-03 | — | — | EP | claimed |
| EP-1675474-B2 | PALATABLE DUCTILE CHEWABLE VETERINARY COMPOSITION | NOVARTIS TIERGESUNDHEIT AG (CH) | 2016-12-07 | — | — | EP | claimed |
| WO-2016001216-A1 | NOVEL METHOD FOR THE TOPICAL APPLICATION OF VETERINARY AGENTS | CEVA SANTE ANIMALE (FR) | 2016-01-07 | — | — | WO | claimed |
| US-20140094418-A1 | PALATABLE DUCTILE CHEWABLE VETERINARY COMPOSITION | NOVARTIS AG (CH) | 2014-04-03 | — | — | US | claimed |
| JP-4754139-B2 | — | — | 2011-08-24 | — | — | JP | claimed |
| US-20090062362-A1 | Veterinary Formulation for Administration of a Water-Insoluble Drug to a Target Animal Through a Water Distribution System | ELANCO ANIMAL HEALTH IRELAND LIMITED (IE) | 2009-03-05 | — | — | US | claimed |
| EP-1675474-B1 | PALATABLE DUCTILE CHEWABLE VETERINARY COMPOSITION | NOVARTIS AG (CH) | 2008-10-22 | — | — | EP | claimed |
| JP-2007500004-A | — | — | 2007-01-11 | — | — | JP | claimed |
| US-20060222684-A1 | Palatable ductile chewable veterinary composition | ELANCO TIERGESUNDHEIT AG (CH) | 2006-10-05 | — | — | US | claimed |
| EP-1675474-A1 | PALATABLE DUCTILE CHEWABLE VETERINARY COMPOSITION | Novartis AG (CH) | 2006-07-05 | — | — | EP | claimed |
| WO-2005013714-A1 | PALATABLE DUCTILE CHEWABLE VETERINARY COMPOSITION | NOVARTIS AG (CH) | 2005-02-17 | — | — | WO | claimed |
| EP-1214052-B1 | VETERINARY FORMULATION FOR ADMINISTRATION OF A WATER-INSOLUBLE DRUG TO A TARGET ANIMAL THROUGH A WATER DISTRIBUTION SYSTEM | JANSSEN PHARMACEUTICA NV (BE) | 2004-08-11 | — | — | EP | claimed |
| EP-1214052-A1 | VETERINARY FORMULATION FOR ADMINISTRATION OF A WATER-INSOLUBLE DRUG TO A TARGET ANIMAL THROUGH A WATER DISTRIBUTION SYSTEM | JANSSEN PHARMACEUTICA N.V. (BE) | 2002-06-19 | — | — | EP | claimed |
| WO-2001017504-A1 | VETERINARY FORMULATION FOR ADMINISTRATION OF A WATER-INSOLUBLE DRUG TO A TARGET ANIMAL THROUGH A WATER DISTRIBUTION SYSTEM | JANSSEN PHARMACEUTICA N.V. (BE) | 2001-03-15 | — | — | WO | claimed |
| EP-0497240-B1 | Preparation for controlled release of drugs for ruminants | HOECHST AG (DE) | 1998-04-08 | — | — | EP | claimed |
| EP-0497240-A1 | Preparation for controlled release of drugs for ruminants | HOECHST AKTIENGESELLSCHAFT (DE) | 1992-08-05 | — | — | EP | claimed |
| EP-0496316-A1 | Pour-on formulation for application of anthelminthics | HOECHST AKTIENGESELLSCHAFT (DE) | 1992-07-29 | — | — | EP | claimed |
| US-11911503-B2 | Manufacturing of semi-plastic pharmaceutical dosage units | INTERVET INC. (US) | 2024-02-27 | — | — | US | disclosed |
| US-20240043446-A1 | ANTHELMINTIC COMPOUNDS COMPRISING A THIENOPYRIDINE STRUCTURE | INTERVET INC. (US) | 2024-02-08 | — | — | US | disclosed |
| US-20240043385-A1 | ANTHELMINTIC COMPOUNDS COMPRISING A PYRIDINE STRUCTURE | INTERVET INC. (US) | 2024-02-08 | — | — | US | disclosed |
| EP-4284509-A1 | ANTIPARASITIC COMPOUNDS | Intervet International B.V. (NL) | 2023-12-06 | — | — | EP | disclosed |
| EP-4153133-B1 | INJECTABLE PHARMACEUTICAL COMPOSITIONS AND USES THEREOF | INTERVET INT BV (NL) | 2023-11-08 | — | — | EP | disclosed |
| US-20230310386-A1 | INJECTABLE PHARMACEUTICAL COMPOSITIONS AND USES THEREOF | INTERVET INC. (US) | 2023-10-05 | — | — | US | disclosed |
| US-20230277448-A1 | CHEWABLE FORMULATIONS | ELANCO TIERGESUNDHEIT AG (CH) | 2023-09-07 | — | — | US | disclosed |
| US-20230263859-A1 | SILK-BASED PRODUCT FORMULATIONS AND METHODS OF USE | COCOON BIOTECH, INC. | 2023-08-24 | — | — | US | disclosed |
| EP-4208155-A1 | CHEWABLE FORMULATIONS | Elanco Tiergesundheit AG (CH) | 2023-07-12 | — | — | EP | disclosed |
| US-20230148316-A1 | ANTHELMINTIC COMPOUNDS COMPRISING A QUINOLINE STRUCTURE | INTERVET INC. (US) | 2023-05-11 | — | — | US | disclosed |
| US-11633455-B2 | Silk-based product formulations and methods of use | COCOON BIOTECH INC. (US) | 2023-04-25 | — | — | US | disclosed |
| CN-111989328-B | Heterocyclic derivatives as pest control agents | 拜耳公司 | 2023-04-18 | — | — | CN | disclosed |
| US-20230110397-A1 | ANTHELMINTIC COMPOUNDS COMPRISING AZAINDOLES STRUCTURE | INTERVET INC. (US) | 2023-04-13 | — | — | US | disclosed |
| CN-112368280-B | Heterocyclic derivatives as pest control agents | 拜耳公司 | 2023-01-20 | — | — | CN | disclosed |
| CN-114929215-A | Palatable soft chews | 礼蓝美国公司 | 2022-08-19 | — | — | CN | disclosed |
| CN-114786484-A | Composition for lice control | 英特维特国际股份有限公司 | 2022-07-22 | — | — | CN | disclosed |
| US-20220218717-A1 | PROCESS FOR MANUFACTURING SOFT CHEWABLE FREE FLOWING GRANULES AND COMPANION ANIMAL PRODUCTS THEREOF | CUCKOS PHARMACEUTICAL PRIVATE LIMITED (IN) | 2022-07-14 | — | — | US | disclosed |
| EP-4025220-A1 | PALATABLE GRANULAR VETERINARY COMPOSITIONS | Elanco US Inc. (US) | 2022-07-13 | — | — | EP | disclosed |
| EP-4025209-A1 | PALATABLE SOFT-CHEW | Elanco US Inc. (US) | 2022-07-13 | — | — | EP | disclosed |
| CN-114727622-A | Palatable granular veterinary compositions | 礼蓝美国公司 | 2022-07-08 | — | — | CN | disclosed |
| US-11337917-B2 | Soft chewable pharmaceutical products | INTERVET INC. (US) | 2022-05-24 | — | — | US | disclosed |
| US-20220142984-A1 | Soft Chewable Pharmaceutical Products | INTERVET INC. (US) | 2022-05-12 | — | — | US | disclosed |
| CN-110382485-B | Heterocyclene derivatives as pest control agents | 拜耳公司 | 2022-05-10 | — | — | CN | disclosed |
| CN-105025885-B | Tablet with improved acceptance and good storage stability | 拜耳动物保健有限责任公司 | 2022-04-08 | — | — | CN | disclosed |
| US-11285101-B2 | Soft chewable pharmaceutical products | INTERVET INC. (US) | 2022-03-29 | — | — | US | disclosed |
| CN-113784702-A | Injectable pharmaceutical composition and use thereof | 英特维特国际股份有限公司 | 2021-12-10 | — | — | CN | disclosed |
| US-20210236420-A1 | Manufacturing of Semi-Plastic Pharmaceutical Dosage Units | INTERVET INC. (US) | 2021-08-05 | — | — | US | disclosed |
| US-20210228684-A1 | SILK-BASED PRODUCT FORMULATIONS AND METHODS OF USE | COCOON BIOTECH INC. | 2021-07-29 | — | — | US | disclosed |
| EP-3393455-B1 | INJECTABLE FORMULATION OF A MACROCYCLIC LACTONE AND LEVAMISOLE | INTERVET INT BV (NL) | 2021-07-21 | — | — | EP | disclosed |
| US-20210177808-A1 | INJECTABLE ISOXAZOLINE PHARMACEUTICAL COMPOSITIONS AND THEIR USE AGAINST PARASITE INFESTATION | INTERVET INC. (US) | 2021-06-17 | — | — | US | disclosed |
| CN-112912377-A | Heterocyclic derivatives as pest control agents | 拜耳公司 | 2021-06-04 | — | — | CN | disclosed |
| US-20210138071-A1 | SILK-BASED PRODUCTS AND METHODS OF USE | COCOON BIOTECH INC. | 2021-05-13 | — | — | US | disclosed |
| US-20210107874-A1 | PHARMACEUTICAL FORMULATION OF CROTONYLAMINOPYRIDINE SALT | INTERVET INC. (US) | 2021-04-15 | — | — | US | disclosed |
| US-10973759-B2 | Manufacturing of semi-plastic pharmaceutical dosage units | INTERVET INC. (US) | 2021-04-13 | — | — | US | disclosed |
| US-20210069104-A1 | PALATABLE SOFT-CHEW | BAYER HEALTHCARE LLC | 2021-03-11 | — | — | US | disclosed |
| US-20210068425-A1 | PALATABLE GRANULAR VETERINARY COMPOSITIONS | BAYER HEALTHCARE LLC | 2021-03-11 | — | — | US | disclosed |
| WO-2021046305-A1 | PALATABLE GRANULAR VETERINARY COMPOSITIONS | BAYER HEALTHCARE LLC (US) | 2021-03-11 | — | — | WO | disclosed |
| WO-2021046296-A1 | PALATABLE SOFT-CHEW | BAYER HEALTHCARE LLC (US) | 2021-03-11 | — | — | WO | disclosed |
| CN-112368280-A | Heterocyclic derivatives as pest control agents | 拜耳公司 | 2021-02-12 | — | — | CN | disclosed |
| WO-2020234898-A1 | PROCESS FOR MANUFACTURING SOFT CHEWABLE FREE FLOWING GRANULES AND COMPANION ANIMAL PRODUCTS THEREOF | CUCKOS PHARMACEUTICAL PRIVATE LIMITED (IO) | 2020-11-26 | — | — | WO | disclosed |
| CN-111989328-A | Heterocyclic derivatives as pest control agents | 拜耳公司 | 2020-11-24 | — | — | CN | disclosed |
| US-10820593-B2 | Methods of preparing alkaloid containing compositions and uses thereof | SYNGENTA PARTICIPATIONS AG (CH) | 2020-11-03 | — | — | US | disclosed |
| US-20200199139-A1 | Alkaloid-Containing Compositions and Uses Thereof | BIOTELLIGA HOLDINGS LIMITED (NZ) | 2020-06-25 | — | — | US | disclosed |
| EP-2627314-B1 | NON-STARCH BASED SOFT CHEWABLES | BAYER IP GMBH (DE) | 2020-05-06 | — | — | EP | disclosed |
| EP-3600300-A1 | PHARMACEUTICAL FORMULATION OF CROTONYLAMINOPYRIDINE SALT | Intervet International B.V. (NL) | 2020-02-05 | — | — | EP | disclosed |
| US-20190336442-A1 | Manufacturing of Semi-Plastic Pharmaceutical Dosage Units | INTERVET INC. (US) | 2019-11-07 | — | — | US | disclosed |
| EP-2831042-B1 | HETEROARYL COMPOUNDS WITH A-CYCLIC BRIDGING UNIT | INTERVET INT BV (NL) | 2019-07-31 | — | — | EP | disclosed |
| US-20190201332-A1 | Soft Chewable Pharmaceutical Products | INTERVET INC. (US) | 2019-07-04 | — | — | US | disclosed |
| US-20190117564-A1 | Soft Chewable Pharmaceutical Products | INTERVET INC. (US) | 2019-04-25 | — | — | US | disclosed |
| US-20190117565-A1 | Soft Chewable Pharmaceutical Product | INTERVET INC. (US) | 2019-04-25 | — | — | US | disclosed |
| EP-1675474-B9 | PALATABLE DUCTILE CHEWABLE VETERINARY COMPOSITION | NOVARTIS TIERGESUNDHEIT AG (CH) | 2018-12-05 | — | — | EP | disclosed |
| EP-2833866-B1 | SOFT CHEWABLE PHARMACEUTICAL PRODUCTS | INTERVET INT BV (NL) | 2018-11-21 | — | — | EP | disclosed |
| EP-3393455-A1 | INJECTABLE FORMULATION OF A MACROCYCLIC LACTONE AND LEVAMISOLE | Intervet International B.V. (NL) | 2018-10-31 | — | — | EP | disclosed |
| WO-2018178345-A1 | PHARMACEUTICAL FORMULATION OF CROTONYLAMINOPYRIDINE SALT | INTERVET INTERNATIONAL B.V. (NL) | 2018-10-04 | — | — | WO | disclosed |
| US-20180280367-A1 | USE OF ANTHELMINTIC AGENTS AGAINST DIROFILARIA IMMITIS | INTERVET INC. (US) | 2018-10-04 | — | — | US | disclosed |
| US-20180263905-A1 | Manufacturing of Semi-Plastic Pharmaceutical Dosage Units | INTERVET INC. (US) | 2018-09-20 | — | — | US | disclosed |
| US-10010538-B2 | Use of anthelmintic agents against Dirofilaria immitis | INTERVET INC. (US) | 2018-07-03 | — | — | US | disclosed |
| CN-105294549-B | N heteroaryl compounds | 英特维特国际股份有限公司 | 2017-12-26 | — | — | CN | disclosed |
| US-20170332641-A1 | METHODS OF PREPARING ALKALOID CONTAINING COMPOSITIONS AND USES THEREOF | SYNGENTA PARTICIPATIONS AG (CH) | 2017-11-23 | — | — | US | disclosed |
| US-20170290766-A1 | SOFT CHEWABLE PHARMACEUTICAL PRODUCTS | INTERVET, INC. (US) | 2017-10-12 | — | — | US | disclosed |
| US-20170266165-A1 | Soft Chewable Pharmaceutical Products | INTERVET INC. (US) | 2017-09-21 | — | — | US | disclosed |
| US-9744127-B2 | Non-starch based soft chewables | BAYER INTELLECTUAL PROPERTY GMBH (DE) | 2017-08-29 | — | — | US | disclosed |
| CN-106998690-A | Process for preparing alkaloid-containing compositions and their use | 先正达参股股份有限公司 | 2017-08-01 | — | — | CN | disclosed |
| US-20170202816-A1 | USE OF ANTHELMINTIC AGENTS AGAINST DIROFILARIA IMMITIS | INTERVET INC. (US) | 2017-07-20 | — | — | US | disclosed |
| US-20170196854-A1 | USE OF ANTHELMINTIC AGENTS AGAINST DIROFILARIA IMMITIS | INTERVET INC. (US) | 2017-07-13 | — | — | US | disclosed |
| WO-2017108954-A1 | INJECTABLE FORMULATION OF A MACROCYCLIC LACTONE AND LEVAMISOLE | INTERVET INTERNATIONAL B.V. (NL) | 2017-06-29 | — | — | WO | disclosed |
| US-20170172918-A1 | SOFT CHEWABLE PHARMACEUTICAL PRODUCTS | INTERVET, INC. (US) | 2017-06-22 | — | — | US | disclosed |
| US-20170172986-A1 | SOFT CHEWABLE PHARMACEUTICAL PRODUCTS | INTERVET, INC. (US) | 2017-06-22 | — | — | US | disclosed |
| US-20170157040-A1 | Manufacturing of Semi-Plastic Pharmaceutical Dosage Units | INTERVET INC. (US) | 2017-06-08 | — | — | US | disclosed |
| US-20170136080-A1 | NOVEL METHOD FOR THE TOPICAL APPLICATION OF VETERINARY AGENTS | Ceva Santé Animale (FR) | 2017-05-18 | — | — | US | disclosed |
| EP-3160506-A1 | NOVEL METHOD FOR THE TOPICAL APPLICATION OF VETERINARY AGENTS | Ceva Sante Animale (FR) | 2017-05-03 | — | — | EP | disclosed |
| US-20170105972-A1 | SOFT CHEWABLE PHARMACEUTICAL PRODUCTS | INTERVET, INC. (US) | 2017-04-20 | — | — | US | disclosed |
| EP-2621923-B1 | N-HETEROARYL COMPOUNDS WITH CYCLIC BRIDGING UNIT FOR THE TREATMENT OF PARASITIC DISEASES | INTERVET INT BV (NL) | 2017-03-29 | — | — | EP | disclosed |
| US-9598412-B2 | Spiroindoline compounds for use as anthelminthics | INTERVET INC. (US) | 2017-03-21 | — | — | US | disclosed |
| EP-2621903-B1 | N-HETEROARYL COMPOUNDS | INTERVET INT BV (NL) | 2017-03-01 | — | — | EP | disclosed |
| US-9532946-B2 | Manufacturing of semi-plastic pharmaceutical dosage units | INTERVET INC. (US) | 2017-01-03 | — | — | US | disclosed |
| EP-1675474-B2 | PALATABLE DUCTILE CHEWABLE VETERINARY COMPOSITION | NOVARTIS TIERGESUNDHEIT AG (CH) | 2016-12-07 | — | — | EP | disclosed |
| EP-2739626-B1 | NOVEL SPIROINDOLINE COMPOUNDS | INTERVET INT BV (NL) | 2016-05-04 | — | — | EP | disclosed |
| US-9321724-B2 | Heteroaryl compounds with A-cyclic bridging unit | INTERVET INC. (US) | 2016-04-26 | — | — | US | disclosed |
| US-9260441-B2 | Heteroaryl compounds with cyclic bridging unit | INTERVET INC. (US) | 2016-02-16 | — | — | US | disclosed |
| CN-105294549-A | N-HETEROARYL COMPOUNDS | INTERVET INT BV | 2016-02-03 | — | — | CN | disclosed |
| WO-2016001216-A1 | NOVEL METHOD FOR THE TOPICAL APPLICATION OF VETERINARY AGENTS | CEVA SANTE ANIMALE (FR) | 2016-01-07 | — | — | WO | disclosed |
| CN-103189356-B | N-heteroaryl compounds | INTERVET INTERNATIONAL B.V. (NL) | 2015-11-25 | — | — | CN | disclosed |
| CN-105025885-A | Tablet with improved acceptance and good storage stability | BAYER ANIMAL HEALTH GMBH | 2015-11-04 | — | — | CN | disclosed |
| US-9096599-B2 | Spiroindoline compounds | INTERVET INC. (US) | 2015-08-04 | — | — | US | disclosed |
| US-9096524-B2 | Anthelmintic agents and their use | INTERVET INTERNATIONAL B.V. (NL) | 2015-08-04 | — | — | US | disclosed |
| US-9040571-B2 | Veterinary formulation for administration of a water-insoluble drug to a target animal through a water distribution system | ELANCO ANIMAL HEALTH IRELAND LIMITED (IE) | 2015-05-26 | — | — | US | disclosed |
| US-20150080365-A1 | HETEROARYL COMPOUNDS WITH CYCLIC BRIDGING UNIT | INTERVET INC. | 2015-03-19 | — | — | US | disclosed |
| US-20150057279-A1 | HETEROARYL COMPOUNDS WITH A-CYCLIC BRIDGING UNIT | INTERVET INC. | 2015-02-26 | — | — | US | disclosed |
| US-20150057302-A1 | SPIROINDOLINE COMPOUNDS FOR USE AS ANTHELMINTHICS | INTERVET INC. | 2015-02-26 | — | — | US | disclosed |
| US-20150057321-A1 | SOFT CHEWABLE PHARMACEUTICAL PRODUCTS | INTERVET INC. | 2015-02-26 | — | — | US | disclosed |
| EP-2830615-A1 | HETEROARYL COMPOUNDS WITH CYCLIC BRIDGING UNIT FOR USE IN THE TREATMENT HELMINTH INFECTION | Intervet International B.V. (NL) | 2015-02-04 | — | — | EP | disclosed |
| EP-2831042-A1 | HETEROARYL COMPOUNDS WITH A-CYCLIC BRIDGING UNIT | Intervet International B.V. (NL) | 2015-02-04 | — | — | EP | disclosed |
| CN-104203214-A | soft chewable pharmaceutical product | INTERVET INT BV | 2014-12-10 | — | — | CN | disclosed |
| US-8883791-B2 | N-heteroaryl compounds with cyclic bridging unit for the treatment of parasitic diseases | INTERVET INC. (US) | 2014-11-11 | — | — | US | disclosed |
| US-8877934-B2 | N-heteroaryl compounds | INTERVET INC. (US) | 2014-11-04 | — | — | US | disclosed |
| EP-2408742-B1 | ANTHELMINTIC AGENTS AND THEIR USE | INTERVET INT BV (NL) | 2014-09-03 | — | — | EP | disclosed |
| EP-2234973-B1 | ANTHELMINTIC AGENTS AND THEIR USE | INTERVET INT BV (NL) | 2014-07-02 | — | — | EP | disclosed |
| US-20140163056-A1 | NOVEL SPIROINDOLINE COMPOUNDS | INTERVET INC. | 2014-06-12 | — | — | US | disclosed |
| US-20140141055-A1 | MANUFACTURING OF SEMI-PLASTIC PHARMACEUTICAL DOSAGE UNITS | INTERVET INC. | 2014-05-22 | — | — | US | disclosed |
| EP-2531506-B1 | Spiroindoline compounds for use as anthelminthics | INTERVET INT BV (NL) | 2014-05-14 | — | — | EP | disclosed |
| US-20140094418-A1 | PALATABLE DUCTILE CHEWABLE VETERINARY COMPOSITION | NOVARTIS AG (CH) | 2014-04-03 | — | — | US | disclosed |
| US-8569495-B2 | Anthelmintic agents and their use | INTERVET INTERNATIONAL B.V. (NL) | 2013-10-29 | — | — | US | disclosed |
| WO-2013144179-A1 | HETEROARYL COMPOUNDS WITH A-CYCLIC BRIDGING UNIT | INTERVET INTERNATIONAL B.V. (NL) | 2013-10-03 | — | — | WO | disclosed |
| WO-2013144180-A1 | HETEROARYL COMPOUNDS WITH CYCLIC BRIDGING UNIT FOR USE IN THE TREATMENT HELMINTH INFECTION | INTERVET INTERNATIONAL B.V. (NL) | 2013-10-03 | — | — | WO | disclosed |
| US-8541019-B2 | Palatable ductile chewable veterinary composition | NOVARTIS AG (CH) | 2013-09-24 | — | — | US | disclosed |
| EP-2627314-A1 | NON-STARCH BASED SOFT CHEWABLES | Bayer Intellectual Property GmbH (DE) | 2013-08-21 | — | — | EP | disclosed |
| US-8507474-B2 | Anthelmintic agents and their use | INTERVET INTERNATIONAL B.V. (NL) | 2013-08-13 | — | — | US | disclosed |
| US-20130203768-A1 | N-HETEROARYL COMPOUNDS WITH CYCLIC BRIDGING UNIT FOR THE TREATMENT OF PARASITIC DISEASES | INTERVET INC. | 2013-08-08 | — | — | US | disclosed |
| EP-2621903-A1 | N-HETEROARYL COMPOUNDS | Intervet International B.V. (NL) | 2013-08-07 | — | — | EP | disclosed |
| EP-2621923-A1 | N-HETEROARYL COMPOUNDS WITH CYCLIC BRIDGING UNIT FOR THE TREATMENT OF PARASITIC DISEASES | Intervet International B.V. (NL) | 2013-08-07 | — | — | EP | disclosed |
| US-20130196993-A1 | N-HETEROARYL COMPOUNDS | INTERVET INC. | 2013-08-01 | — | — | US | disclosed |
| US-20130197006-A1 | Non-Starch Based Soft Chewables | BAYER ANIMAL HEALTH GMBH (DE) | 2013-08-01 | — | — | US | disclosed |
| CN-103200930-A | Non-starch based soft chewables | BAYER IP GMBH | 2013-07-10 | — | — | CN | disclosed |
| CN-103189356-A | N-heteroaryl compounds | INTERVET INT BV | 2013-07-03 | — | — | CN | disclosed |
| EP-2585062-A1 | INJECTABLE FORMULATION OF A MACROCYCLIC LACTONE AND LEVAMISOLE | Intervet International B.V. (NL) | 2013-05-01 | — | — | EP | disclosed |
| US-20130090296-A1 | INJECTABLE FORMULATION OF A MACROCYCLIC LACTONE AND LEVAMISOLE | CHO HYUN SUN (BR) | 2013-04-11 | — | — | US | disclosed |
| EP-2443091-B1 | ANTHELMINTIC AGENTS AND THEIR USE | INTERVET INT BV (NL) | 2013-04-03 | — | — | EP | disclosed |
| EP-2531506-A1 | S PIROINDOLINE COMPOUNDS FOR USE AS ANTHELMINTHI CS | Intervet International B.V. (NL) | 2012-12-12 | — | — | EP | disclosed |
| US-20120295931-A1 | SPIROINDOLINE COMPOUNDS FOR USE AS ANTHELMINTHICS | INTERVET INC. | 2012-11-22 | — | — | US | disclosed |
| EP-2468096-A1 | Anthelmintic combinations | Intervet International BV (NL) | 2012-06-27 | — | — | EP | disclosed |
| EP-2443091-A1 | ANTHELMINTIC AGENTS AND THEIR USE | Intervet International B.V. (NL) | 2012-04-25 | — | — | EP | disclosed |
| US-20120094981-A1 | ANTHELMINTIC AGENTS AND THEIR USE | INTERVET INTERNATIONAL B.V. (NL) | 2012-04-19 | — | — | US | disclosed |
| WO-2012049156-A1 | NON-STARCH BASED SOFT CHEWABLES | BAYER ANIMAL HEALTH GMBH (DE) | 2012-04-19 | — | — | WO | disclosed |
| WO-2012046207-A1 | ANTI-PARASITIC SUBSTITUTED RING FUSED AZINE COMPOUNDS | PARACO TECHNOLOGY LIMITED (NZ) | 2012-04-12 | — | — | WO | disclosed |
| WO-2012041873-A1 | N-HETEROARYL COMPOUNDS | INTERVET INTERNATIONAL B.V. (NL) | 2012-04-05 | — | — | WO | disclosed |
| WO-2012041872-A1 | N-HETEROARYL COMPOUNDS WITH CYCLIC BRIDGING UNIT FOR THE TREATMENT OF PARASITIC DISEASES | INTERVET INTERNATIONAL B.V. (NL) | 2012-04-05 | — | — | WO | disclosed |
| US-20120046296-A1 | PALATABLE DUCTILE CHEWABLE VETERINARY COMPOSITION | ELANCO TIERGESUNDHEIT AG (CH) | 2012-02-23 | — | — | US | disclosed |
| EP-2408742-A1 | ANTHELMINTIC AGENTS AND THEIR USE | Intervet International B.V. (NL) | 2012-01-25 | — | — | EP | disclosed |
| WO-2011161209-A1 | INJECTABLE FORMULATION OF A MACROCYCLIC LACTONE AND LEVAMISOLE | INTERVET INTERNATIONAL B.V. (NL) | 2011-12-29 | — | — | WO | disclosed |
| US-20110319393-A1 | ANTHELMINTIC AGENTS AND THEIR USE | INTERVET INTERNATIONAL B.V. (NL) | 2011-12-29 | — | — | US | disclosed |
| WO-2011095581-A1 | S PIROINDOLINE COMPOUNDS FOR USE AS ANTHELMINTHI CS | INTERVET INTERNATIONAL B.V. (NL) | 2011-08-11 | — | — | WO | disclosed |
| US-20110021506-A1 | ANTHELMINTIC AGENTS AND THEIR USE | INTERVET INTERNATIONAL B.V. (NL) | 2011-01-27 | — | — | US | disclosed |
| WO-2010146083-A1 | ANTHELMINTIC AGENTS AND THEIR USE | INTERVET INTERNATIONAL B.V. (NL) | 2010-12-23 | — | — | WO | disclosed |
| WO-2010115688-A1 | ANTHELMINTIC AGENTS AND THEIR USE | INTERVET INTERNATIONAL B.V. (NL) | 2010-10-14 | — | — | WO | disclosed |
| EP-2234973-A1 | ANTHELMINTIC AGENTS AND THEIR USE | Intervet International B.V. (NL) | 2010-10-06 | — | — | EP | disclosed |
| WO-2009077527-A1 | ANTHELMINTIC AGENTS AND THEIR USE | INTERVET INTERNATIONAL B.V. (NL) | 2009-06-25 | — | — | WO | disclosed |
| US-20090062362-A1 | Veterinary Formulation for Administration of a Water-Insoluble Drug to a Target Animal Through a Water Distribution System | ELANCO ANIMAL HEALTH IRELAND LIMITED (IE) | 2009-03-05 | — | — | US | disclosed |
| WO-2008152081-A2 | ANTHELMINTIC BENZO[D]ISOXAZOLYL BENZAMIDE DERIVATIVES | JANSSEN PHARMACEUTICA NV (BE) | 2008-12-18 | — | — | WO | disclosed |
| US-20080287511-A1 | Anthelmintic Imidazol-Thiazole Derivates | AVISTAR COMMUNICATIONS CORPORATION | 2008-11-20 | — | — | US | disclosed |
| EP-1675474-B1 | PALATABLE DUCTILE CHEWABLE VETERINARY COMPOSITION | NOVARTIS AG (CH) | 2008-10-22 | — | — | EP | disclosed |
| US-20080076703-A1 | Compositions and methods for the enhanced uptake of therapeutic agents through the bladder epithelium | CELL GENESYS, INC. (US) | 2008-03-27 | — | — | US | disclosed |
| US-20060222684-A1 | Palatable ductile chewable veterinary composition | ELANCO TIERGESUNDHEIT AG (CH) | 2006-10-05 | — | — | US | disclosed |
| EP-1675474-A1 | PALATABLE DUCTILE CHEWABLE VETERINARY COMPOSITION | Novartis AG (CH) | 2006-07-05 | — | — | EP | disclosed |
| US-20050059613-A1 | Compositions and methods for the enhanced uptake of therapeutic agents through the bladder epithelium | CELL GENESYS, INC. | 2005-03-17 | — | — | US | disclosed |
| WO-2005013714-A1 | PALATABLE DUCTILE CHEWABLE VETERINARY COMPOSITION | NOVARTIS AG (CH) | 2005-02-17 | — | — | WO | disclosed |
| WO-2005007101-A2 | COMPOSITIONS AND METHODS FOR THE ENHANCED UPTAKE OF THERAPEUTIC AGENTS THROUGH THE BLADDER EPITHELIUM | CELL GENESYS, INC. (US) | 2005-01-27 | — | — | WO | disclosed |
| EP-1214052-B1 | VETERINARY FORMULATION FOR ADMINISTRATION OF A WATER-INSOLUBLE DRUG TO A TARGET ANIMAL THROUGH A WATER DISTRIBUTION SYSTEM | JANSSEN PHARMACEUTICA NV (BE) | 2004-08-11 | — | — | EP | disclosed |
| EP-1237408-B1 | POUR-ON FORMULATIONS | LILLY CO ELI (US) | 2004-02-18 | — | — | EP | disclosed |
| WO-2003051281-A2 | COMPOSITION AND METHOD TO TREAT VIRAL BACTERIAL AND PARASITIC INFECTIONS AND INFESTATIONS | GANADO RESEARCH, L.L.C. (US) | 2003-06-26 | — | — | WO | disclosed |
| EP-1214052-A1 | VETERINARY FORMULATION FOR ADMINISTRATION OF A WATER-INSOLUBLE DRUG TO A TARGET ANIMAL THROUGH A WATER DISTRIBUTION SYSTEM | JANSSEN PHARMACEUTICA N.V. (BE) | 2002-06-19 | — | — | EP | disclosed |
| WO-2001017504-A1 | VETERINARY FORMULATION FOR ADMINISTRATION OF A WATER-INSOLUBLE DRUG TO A TARGET ANIMAL THROUGH A WATER DISTRIBUTION SYSTEM | JANSSEN PHARMACEUTICA N.V. (BE) | 2001-03-15 | — | — | WO | disclosed |
| EP-0497240-B1 | Preparation for controlled release of drugs for ruminants | HOECHST AG (DE) | 1998-04-08 | — | — | EP | disclosed |
| EP-0497240-A1 | Preparation for controlled release of drugs for ruminants | HOECHST AKTIENGESELLSCHAFT (DE) | 1992-08-05 | — | — | EP | disclosed |
| EP-0496316-A1 | Pour-on formulation for application of anthelminthics | HOECHST AKTIENGESELLSCHAFT (DE) | 1992-07-29 | — | — | EP | disclosed |
| EP-0496316-A1 | Pour-on formulation for application of anthelminthics | HOECHST AKTIENGESELLSCHAFT (DE) | 1992-07-29 | — | — | EP | disclosed |
| EP-0496316-A1 | Pour-on formulation for application of anthelminthics | HOECHST AKTIENGESELLSCHAFT (DE) | 1992-07-29 | — | — | EP | disclosed |
Patent text — is the patent's own abstract consistent with the prediction?
For each of this compound's patents that has machine-readable text (50 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.
| Patent | Title | Text reads most about | Predicted target · text-rank |
|---|---|---|---|
| US-20210177808-A1 | INJECTABLE ISOXAZOLINE PHARMACEUTICAL COMPOSITIONS AND THEIR USE AGAINST PARASITE INFESTATION | INA, MMP1, EPX | ELANE 437/4885FAAH 2695/4885AURKA 4519/4885 |
| US-20110021506-A1 | ANTHELMINTIC AGENTS AND THEIR USE | ACHE, ABCB11, MPO | ELANE 113/4885FAAH 228/4885AURKA 1046/4885 |
| US-20110319393-A1 | ANTHELMINTIC AGENTS AND THEIR USE | ACHE, ABCB11, MPO | ELANE 113/4885FAAH 228/4885AURKA 1046/4885 |
| US-20180263905-A1 | Manufacturing of Semi-Plastic Pharmaceutical Dosage Units | PUF60, RPS11, RPS20 | ELANE 4476/4885FAAH 4017/4885AURKA 4249/4885 |
| US-20170157040-A1 | Manufacturing of Semi-Plastic Pharmaceutical Dosage Units | PUF60, RPS11, RPS20 | ELANE 4476/4885FAAH 4017/4885AURKA 4249/4885 |
| US-20050059613-A1 | Compositions and methods for the enhanced uptake of therapeutic agents through the bladder epithelium | MUC1, SLC17A5, CD44 | ELANE 218/4885FAAH 3611/4885AURKA 4871/4885 |
| US-20140141055-A1 | MANUFACTURING OF SEMI-PLASTIC PHARMACEUTICAL DOSAGE UNITS | PUF60, RPS11, RPS20 | ELANE 4476/4885FAAH 4017/4885AURKA 4249/4885 |
| US-20150057321-A1 | SOFT CHEWABLE PHARMACEUTICAL PRODUCTS | PAM, TAS2R46, TAS2R16 | ELANE 3486/4885FAAH 1769/4885AURKA 2932/4885 |
| US-20060222684-A1 | Palatable ductile chewable veterinary composition | PIGO, TAS2R41, TAS2R30 | ELANE 59/4885FAAH 2217/4885AURKA 4264/4885 |
| US-20220142984-A1 | Soft Chewable Pharmaceutical Products | PAM, TAS2R46, TAS2R16 | ELANE 3486/4885FAAH 1769/4885AURKA 2932/4885 |
| US-10973759-B2 | Manufacturing of semi-plastic pharmaceutical dosage units | PUF60, RPS11, RPS20 | ELANE 4476/4885FAAH 4017/4885AURKA 4249/4885 |
| US-20210236420-A1 | Manufacturing of Semi-Plastic Pharmaceutical Dosage Units | PUF60, RPS11, RPS20 | ELANE 4476/4885FAAH 4017/4885AURKA 4249/4885 |
| US-20080076703-A1 | Compositions and methods for the enhanced uptake of therapeutic agents through the bladder epithelium | MUC1, SLC17A5, CD44 | ELANE 218/4885FAAH 3611/4885AURKA 4871/4885 |
| US-20170332641-A1 | METHODS OF PREPARING ALKALOID CONTAINING COMPOSITIONS AND USES THEREOF | INMT, LSS, ACHE | ELANE 3094/4885FAAH 1900/4885AURKA 3146/4885 |
| US-11911503-B2 | Manufacturing of semi-plastic pharmaceutical dosage units | PUF60, RPS11, RPS20 | ELANE 4476/4885FAAH 4017/4885AURKA 4249/4885 |
| US-20150080365-A1 | HETEROARYL COMPOUNDS WITH CYCLIC BRIDGING UNIT | PIGS, MTCL3, GJB2 | ELANE 842/4885FAAH 294/4885AURKA 1894/4885 |
| US-11285101-B2 | Soft chewable pharmaceutical products | PAM, TAS2R46, TAS2R16 | ELANE 3486/4885FAAH 1769/4885AURKA 2932/4885 |
| US-20240043385-A1 | ANTHELMINTIC COMPOUNDS COMPRISING A PYRIDINE STRUCTURE | HRH4, PNPO, NME4 | ELANE 416/4885FAAH 315/4885AURKA 2252/4885 |
| US-20150057279-A1 | HETEROARYL COMPOUNDS WITH A-CYCLIC BRIDGING UNIT | AADAC, PIGS, MTCL3 | ELANE 1585/4885FAAH 270/4885AURKA 506/4885 |
| US-20230277448-A1 | CHEWABLE FORMULATIONS | SI, TAS2R39, TAS2R31 | ELANE 3089/4885FAAH 1288/4885AURKA 1989/4885 |
| US-20150057302-A1 | SPIROINDOLINE COMPOUNDS FOR USE AS ANTHELMINTHICS | PKD2, PKD1, PIR | ELANE 1955/4885FAAH 1080/4885AURKA 2533/4885 |
| US-20130196993-A1 | N-HETEROARYL COMPOUNDS | HNMT, SQLE, PIGO | ELANE 245/4885FAAH 192/4885AURKA 2761/4885 |
| US-20170290766-A1 | SOFT CHEWABLE PHARMACEUTICAL PRODUCTS | PAM, TAS2R46, TAS2R16 | ELANE 3486/4885FAAH 1769/4885AURKA 2932/4885 |
| US-20170196854-A1 | USE OF ANTHELMINTIC AGENTS AGAINST DIROFILARIA IMMITIS | MPO, DHODH, DHX35 | ELANE 8/4885FAAH 314/4885AURKA 2641/4885 |
| US-20180280367-A1 | USE OF ANTHELMINTIC AGENTS AGAINST DIROFILARIA IMMITIS | MPO, DHODH, DHX35 | ELANE 8/4885FAAH 314/4885AURKA 2641/4885 |
| US-20210069104-A1 | PALATABLE SOFT-CHEW | TAS2R40, TAS2R45, TAS2R42 | ELANE 261/4885FAAH 95/4885AURKA 4639/4885 |
| US-20190117564-A1 | Soft Chewable Pharmaceutical Products | PAM, TAS2R46, TAS2R16 | ELANE 3486/4885FAAH 1769/4885AURKA 2932/4885 |
| US-20170266165-A1 | Soft Chewable Pharmaceutical Products | PAM, TAS2R46, TAS2R16 | ELANE 3486/4885FAAH 1769/4885AURKA 2932/4885 |
| US-10010538-B2 | Use of anthelmintic agents against Dirofilaria immitis | MPO, DHODH, DHX35 | ELANE 8/4885FAAH 314/4885AURKA 2641/4885 |
| US-10820593-B2 | Methods of preparing alkaloid containing compositions and uses thereof | LSS, LARP7, ACHE | ELANE 3638/4885FAAH 1910/4885AURKA 1934/4885 |
| US-20190117565-A1 | Soft Chewable Pharmaceutical Product | PAM, TAS2R46, TAS2R16 | ELANE 3541/4885FAAH 1773/4885AURKA 2803/4885 |
| US-20120295931-A1 | SPIROINDOLINE COMPOUNDS FOR USE AS ANTHELMINTHICS | PKD2, PKD1, PIR | ELANE 1955/4885FAAH 1080/4885AURKA 2533/4885 |
| US-20240043446-A1 | ANTHELMINTIC COMPOUNDS COMPRISING A THIENOPYRIDINE STRUCTURE | DHODH, NISCH, DDT | ELANE 570/4885FAAH 272/4885AURKA 2450/4885 |
| US-20130203768-A1 | N-HETEROARYL COMPOUNDS WITH CYCLIC BRIDGING UNIT FOR THE TREATMENT OF PARASITIC DISEASES | PIGO, HNMT, PIGS | ELANE 609/4885FAAH 331/4885AURKA 2331/4885 |
| US-20080287511-A1 | Anthelmintic Imidazol-Thiazole Derivates | NOD1, IL33, IL5 | ELANE 39/4885FAAH 492/4885AURKA 630/4885 |
| US-20230148316-A1 | ANTHELMINTIC COMPOUNDS COMPRISING A QUINOLINE STRUCTURE | DHX35, DDX5, DHODH | ELANE 109/4885FAAH 270/4885AURKA 2325/4885 |
| US-20210107874-A1 | PHARMACEUTICAL FORMULATION OF CROTONYLAMINOPYRIDINE SALT | SUCNR1, SLC5A2, CS | ELANE 4136/4885FAAH 4642/4885AURKA 4236/4885 |
| US-20230310386-A1 | INJECTABLE PHARMACEUTICAL COMPOSITIONS AND USES THEREOF | CYP3A7, PDE8A, CYP4X1 | ELANE 2016/4885FAAH 4688/4885AURKA 3189/4885 |
| US-20210068425-A1 | PALATABLE GRANULAR VETERINARY COMPOSITIONS | PIGS, VMA21, PGA5 | ELANE 1352/4885FAAH 1050/4885AURKA 4479/4885 |
| US-20170105972-A1 | SOFT CHEWABLE PHARMACEUTICAL PRODUCTS | PAM, TAS2R46, TAS2R16 | ELANE 3486/4885FAAH 1769/4885AURKA 2932/4885 |
| US-20230110397-A1 | ANTHELMINTIC COMPOUNDS COMPRISING AZAINDOLES STRUCTURE | AADAC, HNMT, NISCH | ELANE 97/4885FAAH 254/4885AURKA 1663/4885 |
| US-11337917-B2 | Soft chewable pharmaceutical products | PAM, TAS2R46, TAS2R16 | ELANE 3486/4885FAAH 1769/4885AURKA 2932/4885 |
| US-20170202816-A1 | USE OF ANTHELMINTIC AGENTS AGAINST DIROFILARIA IMMITIS | MPO, DHODH, DHX35 | ELANE 8/4885FAAH 314/4885AURKA 2641/4885 |
| US-20140163056-A1 | NOVEL SPIROINDOLINE COMPOUNDS | PKD2, PKD1, REN | ELANE 2327/4885FAAH 1112/4885AURKA 2964/4885 |
| US-20200199139-A1 | Alkaloid-Containing Compositions and Uses Thereof | ACHE, TAC3, LARP7 | ELANE 3446/4885FAAH 2180/4885AURKA 1495/4885 |
| US-20170172918-A1 | SOFT CHEWABLE PHARMACEUTICAL PRODUCTS | PAM, TAS2R46, TAS2R16 | ELANE 3486/4885FAAH 1769/4885AURKA 2932/4885 |
| US-20190201332-A1 | Soft Chewable Pharmaceutical Products | PAM, TAS2R46, TAS2R16 | ELANE 3486/4885FAAH 1769/4885AURKA 2932/4885 |
| US-20190336442-A1 | Manufacturing of Semi-Plastic Pharmaceutical Dosage Units | PUF60, RPS11, RPS20 | ELANE 4476/4885FAAH 4017/4885AURKA 4249/4885 |
| US-20120094981-A1 | ANTHELMINTIC AGENTS AND THEIR USE | ABCB11, ACHE, CMA1 | ELANE 137/4885FAAH 51/4885AURKA 920/4885 |
| US-20170172986-A1 | SOFT CHEWABLE PHARMACEUTICAL PRODUCTS | PAM, TAS2R46, TAS2R16 | ELANE 3486/4885FAAH 1769/4885AURKA 2932/4885 |
“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.