SCHEMBL4565426

SCHEMBL4565426

CNc1ccnc2cc(-c3ccc(S(=O)(=O)C4CCC5(CC4)CC(C4CC4)C(=O)CN5)cc3)ccc12

nearest known ligand 0.38

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
TGFBR1 P36897 13/20 0.38
MAP4K4 O95819 8/20 0.38
PIK3C3 Q8NEB9 1/20 0.33
ALK Q9UM73 4/20 0.31
CCR7 P32248 1/20 0.31
CCR6 P51684 1/20 0.31
LRRK2 Q5S007 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4565595 0.88 KCNH2 (0.34) TGFBR1MAP4K4PIK3C3ALK
SCHEMBL4565379 0.86 IRAK4 (0.34) PIK3C3ALK
SCHEMBL4565577 0.78 SGK1 (0.46)
SCHEMBL4565605 0.75 MAPK14 (0.37)
SCHEMBL4564596 0.75 CD74 (0.34) CCR6
SCHEMBL4564399 0.75 FASN (0.37) CCR6
SCHEMBL4565405 0.75 PTGER3 (0.34)
SCHEMBL4565553 0.75 FGFR1 (0.37) MAP4K4
SCHEMBL4564364 0.74 HTR6 (0.36)
SCHEMBL4536541 0.74

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2637660-A1 FATTY ACID SYNTHASE INHIBITORS Glaxosmithkline Intellectual Property (No. 2) Limited (GB) 2013-09-18 EP disclosed
WO-2012064642-A1 FATTY ACID SYNTHASE INHIBITORS GLAXOSMITHKLINE LLC (US) 2012-05-18 WO disclosed