SCHEMBL456774

SCHEMBL456774

Cc1cc(Cl)c(N2CCN(C(C)(C)C)CC2)cc1NC(=O)OC(C)(C)C

nearest known ligand 0.40

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
DRD2 P14416 4/20 0.36
LMNA P02545 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
BACE1 P56817 2/20 0.36
XPO1 O14980 1/20 0.35
ATR Q13535 1/20 0.35
LCK P06239 2/20 0.35
DRD3 P35462 1/20 0.35
NPY2R P49146 2/20 0.34
NPC1 O15118 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12457410 0.88 KDM4E (0.41) MEN1KMT2ALMNANPSR1NPY2R
SCHEMBL457432 0.87 MEN1 (0.51) MEN1KMT2ALMNANPSR1BACE1
SCHEMBL459024 0.80 LMNA (0.43) MEN1KMT2ALMNANPSR1
SCHEMBL470212 0.78 MEN1 (0.51) MEN1KMT2ALMNANPSR1BACE1
SCHEMBL458554 0.77 NPY2R (0.42) MEN1KMT2ALMNABACE1NPY2R
SCHEMBL470197 0.77 MEN1 (0.47) MEN1KMT2ALMNANPSR1BACE1
SCHEMBL470229 0.76 MEN1 (0.46) MEN1KMT2ALMNANPSR1BACE1
SCHEMBL6164833 0.76 KDM4E (0.41) MEN1KMT2ALMNANPSR1NPC1
SCHEMBL6166440 0.76 KDM4E (0.39) MEN1KMT2ADRD2LMNANPSR1
SCHEMBL15414721 0.75 GPR35 (0.40) DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2614052-A1 NOVEL PIPERAZINE ANALOGS AS BROAD-SPECTRUM INFLUENZA ANTIVIRALS Bristol-Myers Squibb Company (US) 2013-07-17 EP disclosed
WO-2012033736-A1 NOVEL PIPERAZINE ANALOGS AS BROAD-SPECTRUM INFLUENZA ANTIVIRALS BRISTOL-MYERS SQUIBB COMPANY (US) 2012-03-15 WO disclosed