SCHEMBL4569732

SCHEMBL4569732

CCOc1c(OC[C@H]2CO2)ccc2c1N=C(N)N1CCN=C21

nearest known ligand 0.34

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.34
GLA P06280 1/20 0.34
HRH3 Q9Y5N1 3/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
CA4 P22748 1/20 0.33
CA7 P43166 1/20 0.33
KMT2A Q03164 3/20 0.32
MEN1 O00255 2/20 0.31
TP53 P04637 2/20 0.30
MAPT P10636 2/20 0.30
HPGD P15428 2/20 0.30
TSHR P16473 2/20 0.30
CYP1A2 P05177 1/20 0.30
PPARG P37231 1/20 0.30
HIF1A Q16665 1/20 0.30
DRD4 P21917 2/20 0.30
VDR P11473 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4532060 0.91 PTAFR (0.35) ALDH1A1GLACA1CA2CA4
SCHEMBL4539391 0.91 PTAFR (0.35) ALDH1A1GLACA1CA2CA4
SCHEMBL4529772 0.91 PTAFR (0.35) ALDH1A1GLACA1CA2CA4
SCHEMBL18928155 0.76 PTAFR (0.36) CA1CA2CA4CA7
SCHEMBL30137694 0.71 PTAFR (0.41) ALDH1A1KMT2AMEN1TSHR
SCHEMBL1655758 0.71 PTAFR (0.41) ALDH1A1KMT2AMEN1TSHR
SCHEMBL12362314 0.70 HDAC8 (0.39) CA1CA2CA4CA7
SCHEMBL4569733 0.70 ALDH1A1 (0.38) ALDH1A1KMT2AMEN1MAPTHPGD
SCHEMBL17732339 0.70 P2RX7 (0.34) ALDH1A1TP53MAPTHPGDTSHR
SCHEMBL1658299 0.69 KDM4E (0.41) ALDH1A1KMT2AMEN1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2638043-A1 ARYLAMINOALCOHOL-SUBSTITUTED 2,3-DIHYDROIMIDAZO[1,2-C]QUINOLINES Bayer Intellectual Property GmbH (DE) 2013-09-18 EP disclosed
WO-2012062743-A1 ARYLAMINOALCOHOL-SUBSTITUTED 2,3-DIHYDROIMIDAZO[1,2-C]QUINOLINES BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2012-05-18 WO disclosed