SCHEMBL456995

SCHEMBL456995

Cc1[c]c(Br)ccc1-c1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.41
MAPK1 P28482 2/20 0.41
ESR2 Q92731 1/20 0.38
CYP2A6 P11509 2/20 0.36
CYP2B6 P20813 1/20 0.36
AKT1 P31749 1/20 0.34
AKT2 P31751 1/20 0.34
BACE1 P56817 1/20 0.33
ALOX5 P09917 1/20 0.33
PDCD1 Q15116 1/20 0.33
CD274 Q9NZQ7 1/20 0.33
LMNA P02545 3/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
MCOLN3 Q8TDD5 2/20 0.33
KDM4E B2RXH2 2/20 0.33
MAPT P10636 1/20 0.33
NR2F2 P24468 1/20 0.33
HTT P42858 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
HSD17B10 Q99714 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4371389 0.78 ESR2 (0.41) ALDH1A1MAPK1ESR2CYP2A6CYP2B6
SCHEMBL457364 0.78 ALDH1A1 (0.44) ALDH1A1MAPK1ESR2CYP2A6BACE1
SCHEMBL27714313 0.75 ESR2 (0.47) ALDH1A1ESR2CYP2A6CYP2B6AKT1
SCHEMBL6206554 0.75 CYP2A6 (0.41) ALDH1A1ESR2CYP2A6CYP2B6AKT1
SCHEMBL456919 0.75 ALDH1A1 (0.41) ALDH1A1MAPK1ESR2CYP2A6BACE1
SCHEMBL456233 0.75 ESR2 (0.38) ALDH1A1MAPK1ESR2CYP2A6CYP2B6
SCHEMBL455577 0.75 ALDH1A1 (0.41) ALDH1A1MAPK1ESR2CYP2A6BACE1
SCHEMBL455612 0.75 ALDH1A1 (0.38) ALDH1A1MAPK1BACE1LMNASMN1; SMN2
SCHEMBL28926395 0.73 BACE1 (0.44) ALDH1A1MAPK1ESR2CYP2A6CYP2B6
SCHEMBL457524 0.71 ALDH1A1 (0.41) ALDH1A1MAPK1ESR2CYP2A6CYP2B6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2614053-A1 METHOD FOR PRODUCING PYRIDAZINONE COMPOUNDS AND INTERMEDIATE THEREOF SUMITOMO CHEMICAL COMPANY LIMITED (JP) 2013-07-17 EP disclosed
WO-2012033225-A1 METHOD FOR PRODUCING PYRIDAZINONE COMPOUNDS AND INTERMEDIATE THEREOF SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2012-03-15 WO disclosed