SCHEMBL455612

SCHEMBL455612

COc1[c]c(Br)ccc1-c1ccccc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.38
MAPK1 P28482 1/20 0.38
SQOR Q9Y6N5 2/20 0.34
BACE1 P56817 2/20 0.34
PTPN1 P18031 1/20 0.34
NPSR1 Q6W5P4 2/20 0.34
LMNA P02545 1/20 0.34
POLB P06746 1/20 0.34
PDE4B Q07343 3/20 0.33
MAPT P10636 3/20 0.33
HTT P42858 2/20 0.33
NCOA1 Q15788 1/20 0.33
NCOA3 Q9Y6Q9 1/20 0.33
MAOB P27338 1/20 0.33
MITF O75030 1/20 0.33
PDE4A P27815 1/20 0.33
PDE4C Q08493 1/20 0.33
PDE4D Q08499 1/20 0.33
CA4 P22748 1/20 0.32
NPC1 O15118 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL456629 0.79 SQOR (0.39) ALDH1A1SQORBACE1NPSR1PDE4B
SCHEMBL7820403 0.79 PDE4B (0.38) ALDH1A1MAPK1SQORBACE1NPSR1
SCHEMBL8548982 0.79 APP (0.42) ALDH1A1PTPN1NPSR1LMNAMAPT
SCHEMBL458401 0.78 SQOR (0.34) ALDH1A1SQORBACE1PTPN1NPSR1
SCHEMBL457574 0.78 SQOR (0.38) ALDH1A1SQORBACE1NPSR1POLB
SCHEMBL21331773 0.76 BACE1 (0.42) ALDH1A1SQORBACE1NPSR1PDE4B
SCHEMBL456995 0.75 ALDH1A1 (0.41) ALDH1A1MAPK1BACE1NPSR1LMNA
SCHEMBL457364 0.74 ALDH1A1 (0.44) ALDH1A1MAPK1BACE1MAPTRAB9A
SCHEMBL457181 0.73 ADRB2 (0.33) ALDH1A1MAPK1SQORBACE1NPSR1
SCHEMBL455577 0.71 ALDH1A1 (0.41) ALDH1A1MAPK1BACE1LMNAHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2614053-A1 METHOD FOR PRODUCING PYRIDAZINONE COMPOUNDS AND INTERMEDIATE THEREOF SUMITOMO CHEMICAL COMPANY LIMITED (JP) 2013-07-17 EP disclosed
WO-2012033225-A1 METHOD FOR PRODUCING PYRIDAZINONE COMPOUNDS AND INTERMEDIATE THEREOF SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2012-03-15 WO disclosed