SCHEMBL4570033

SCHEMBL4570033

Fc1ccccc1C(F)Oc1ccc(Br)cc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LDHA P00338 1/20 0.38
SLC6A4 P31645 1/20 0.36
IDO1 P14902 2/20 0.35
TDO2 P48775 2/20 0.35
MEN1 O00255 3/20 0.34
KMT2A Q03164 3/20 0.34
IGLV6-57 P01721 1/20 0.32
ALDH1A1 P00352 3/20 0.32
MAPT P10636 5/20 0.32
CES2 O00748 2/20 0.32
CES1 P23141 2/20 0.32
LMNA P02545 2/20 0.32
NPC1 O15118 1/20 0.32
HTT P42858 1/20 0.32
RAB9A P51151 1/20 0.32
KDM4E B2RXH2 2/20 0.31
POLB P06746 1/20 0.31
CNR2 P34972 1/20 0.31
L3MBTL1 Q9Y468 2/20 0.31
PKM P14618 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18094440 0.78 LDHA (0.35) LDHASLC6A4IDO1TDO2MEN1
SCHEMBL28869187 0.76 SLC6A4 (0.49) LDHASLC6A4MEN1KMT2AALDH1A1
SCHEMBL5140182 0.72 IDO1 (0.44) SLC6A4IDO1TDO2MEN1KMT2A
SCHEMBL16111990 0.70 IGF1R (0.42) SLC6A4IDO1TDO2MEN1KMT2A
SCHEMBL157708 0.69 ALOX15 (0.50) LDHASLC6A4MEN1KMT2AALDH1A1
SCHEMBL327420 0.69 IDO1 (0.51) SLC6A4IDO1TDO2MEN1KMT2A
SCHEMBL9729013 0.67 HTR2A (0.41) IDO1TDO2MEN1KMT2AALDH1A1
SCHEMBL16111744 0.67 HTR2A (0.37) IDO1TDO2MEN1KMT2AALDH1A1
SCHEMBL7766235 0.66 LDHA (0.47) LDHASLC6A4MEN1KMT2AALDH1A1
SCHEMBL28384768 0.66 LDHA (0.47) LDHASLC6A4MEN1KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2117535-A1 NOVEL PHARMACEUTICAL COMPOSITIONS Glaxo Group Limited (GB) 2009-11-18 EP disclosed
WO-2008090116-A1 NOVEL PHARMACEUTICAL COMPOSITIONS GLAXO GROUP LIMITED (GB) 2008-07-31 WO disclosed