SCHEMBL457065

SCHEMBL457065

COc1cc(N=C=S)cc(OC)c1OC

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACHE P22303 1/20 0.46
CYP3A4 P08684 2/20 0.45
MAPT P10636 2/20 0.45
CA9 Q16790 1/20 0.45
PTGS2 P35354 1/20 0.42
CYP1A1 P04798 2/20 0.40
CYP1B1 Q16678 2/20 0.40
HPGD P15428 3/20 0.39
ALDH1A1 P00352 3/20 0.39
KDM4E B2RXH2 2/20 0.39
CYP1A2 P05177 2/20 0.39
CYP2D6 P10635 1/20 0.39
G6PD P11413 1/20 0.39
CYP2C9 P11712 1/20 0.39
PKM P14618 1/20 0.39
ALOX15 P16050 1/20 0.39
ALOX12 P18054 1/20 0.39
HK1 P19367 1/20 0.39
CYP2C19 P33261 1/20 0.39
MPI P34949 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23760097 0.82 GAA (0.46) CYP3A4MAPTCA9PTGS2HPGD
SCHEMBL11382490 0.81 KDM4E (0.48) MAPTHPGDALDH1A1KDM4EPKM
SCHEMBL11393184 0.81 HTT (0.41) MAPTHPGDALDH1A1KDM4EAPOBEC3G
SCHEMBL374491 0.79 CYP3A4 (0.47) ACHECYP3A4MAPTCA9PTGS2
SCHEMBL11383026 0.78 PDE3B (0.41) CYP3A4MAPTALDH1A1KDM4ETUBB4A
SCHEMBL11383070 0.78 ALDH1A1 (0.43) MAPTPTGS2HPGDALDH1A1KDM4E
SCHEMBL76835 0.78 HTR3E (0.53) ACHECYP3A4MAPTCA9PTGS2
SCHEMBL1119953 0.77 NAAA (0.35) TUBB1
SCHEMBL6179404 0.75 P2RY6 (0.38) CYP3A4MAPTPTGS2HPGDALDH1A1
SCHEMBL1021008 0.74 ALDH1A1 (0.50) CYP3A4MAPTCA9PTGS2CYP1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 138 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20160250175-A1 COMBINED APPLICATION OF ISOTHIOCYANATE COMPOUND AND ANTI-CANCER MEDICINE JC (WUXI) COMPANY, INC. (CN) 2016-09-01 US claimed
EP-3034076-A1 COMBINED APPLICATION OF ISOTHIOCYANATE COMPOUND AND ANTI-CANCER MEDICINE JC (Wuxi) COMPANY, Inc. (CN) 2016-06-22 EP claimed
CN-105267967-A Combined application of isothiocyanate-type compound and anti-cancer drug acting or affecting DNA WUXI JC PHARMACAUTICAL TECHNOLOGY INC 2016-01-27 CN claimed
CN-104415332-A Combined application between isothiocyanate-type compound and kinase inhibitor medicine in treatment of cancer WUXI JC PHARMACAUTICAL TECHNOLOGY INC 2015-03-18 CN claimed
CN-104117064-A Combined application of isothiocyanate compound and hormone medicine WUXI JC PHARMACAUTICAL TECHNOLOGY INC 2014-10-29 CN claimed
EP-3446689-B1 ISOTHIOCYANATE COMPOUND FOR USE IN THE TREATMENT OF HYPERBILIRUBINEMIA JC WUXI COMPANY INC (CN) 2025-01-08 EP disclosed
CN-118873522-A Application of isothiocyanate compound 无锡杰西医药股份有限公司 2024-11-01 CN disclosed
CN-118619952-A Aloperine derivative, preparation method, pharmaceutical composition and application thereof 中国医学科学院药物研究所 2024-09-10 CN disclosed
CN-113262218-B Use of isothiocyanate compounds 无锡杰西医药股份有限公司 2024-06-18 CN disclosed
CN-114540846-B Synthesis method of 1,2, 4-triazolo six-membered nitrogen heterocycle-3-amine 五邑大学 2023-09-19 CN disclosed
CN-114516870-B Triazolo hexa-nitrogen heterocyclic-3-amine compound and preparation method and application thereof 五邑大学 2023-04-11 CN disclosed
CN-113354592-B 2-thioquinazolinone compound and preparation method and application thereof 赣南师范大学 2022-06-21 CN disclosed
US-5246935-A Cardiovascular and gastrointestinal NOVO NORDISK A/S (DK) 1993-09-21 US disclosed
EP-0544765-A1 PIPERAZINYL DERIVATIVES. NOVO NORDISK AS (DK) 1993-06-09 EP disclosed
CN-1069490-A Urea derivatives YAMANOUCHI PHARMA CO LTD (JP) 1993-03-03 CN disclosed
US-5190961-A Bactericides TERUMO KABUSHIKI KAISHA (JP) 1993-03-02 US disclosed
WO-1992003426-A1 PIPERAZINYL DERIVATIVES NOVO NORDISK A/S (DK) 1992-03-05 WO disclosed
EP-0470006-A1 Thiourea derivatives and antimicrobial agent and antiulcer agent containing the same TERUMO KABUSHIKI KAISHA (JP) 1992-02-05 EP disclosed
US-4634660-A ANTIFOGGING AGENT FUJI PHOTO FILM CO., LTD. (JP) 1987-01-06 US disclosed
EP-0123146-A2 Compound with antiinflammatory activity, process for preparation thereof and pharmaceutical compositions therefrom CHIESI FARMACEUTICI S.p.A. (IT) 1984-10-31 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20160250175-A1 COMBINED APPLICATION OF ISOTHIOCYANATE COMPOUND AND ANTI-CANCER MEDICINE CHUK, KIT, MKI67 ACHE 1947/4885CYP3A4 2452/4885MAPT 4080/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.