Tromethamine

Tromethamine

SCHEMBL457183

Bc1c(F)c(F)c(F)c(F)c1F.NC(CO)(CO)CO

nearest known ligand 0.50

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

DHFRGARTPTGFRPTGIRPTGS1PTGS2TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBBTUBB1TUBB2ATUBB2BTUBB3TUBB4ATUBB4BTUBB6TUBB8envmurAthyA

The experimentally established mechanism targets of Tromethamine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.50
LMNA P02545 1/20 0.50
KMT2A Q03164 1/20 0.50
S1PR1 P21453 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Tromethamine SCHEMBL6864894 0.98 MEN1 (0.48) MEN1LMNAKMT2A
Tromethamine SCHEMBL8618035 0.88 MEN1 (0.39) MEN1LMNAKMT2A
Tromethamine SCHEMBL8616153 0.87 MEN1 (0.42) MEN1LMNAKMT2A
Tromethamine SCHEMBL7028618 0.83 MEN1 (0.34) MEN1LMNAKMT2A
Tromethamine SCHEMBL9193688 0.82 MEN1 (0.42) MEN1LMNAKMT2AS1PR1
Tromethamine SCHEMBL19856508 0.75 MEN1 (0.50) MEN1LMNAKMT2AS1PR1
Tromethamine SCHEMBL16702277 0.75 MEN1 (0.50) MEN1LMNAKMT2AS1PR1
Tromethamine SCHEMBL18729667 0.75 MEN1 (0.50) MEN1LMNAKMT2AS1PR1
Tromethamine SCHEMBL8531348 0.73 MEN1 (0.42) MEN1LMNAKMT2AS1PR1
Tromethamine SCHEMBL7652452 0.73 MEN1 (0.42) MEN1LMNAKMT2AS1PR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 113 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20020183574-A1 Hydrocarbon conversion process SASOL TECHNOLOGY (PTY) LTD. (ZA) 2002-12-05 US claimed
EP-1235767-A1 HYDROCARBON CONVERSION PROCESS Sasol Technology (Proprietary) Limited (ZA) 2002-09-04 EP claimed
WO-2002038637-A1 METHOD FOR COPOLYMERIZING PROPENE AND/OR ETHENE WITH 1-OLEFINS ON METALLOCENE CARRIER CATALYSTS BASELL POLYPROPYLEN GMBH (DE) 2002-05-16 WO claimed
WO-2001038270-A1 HYDROCARBON CONVERSION PROCESS SASOL TECHNOLOGY (PTY) LTD (ZA) 2001-05-31 WO claimed
EP-0632819-B1 ADDITION POLYMERIZATION CATALYSTS COMPRISING REDUCED OXIDATION STATE METAL COMPLEXES DOW CHEMICAL CO (US) 1998-09-02 EP claimed
EP-3066140-B1 STEREOREGULAR DIBLOCK POLYBUTADIENES HAVING A 1,4-CIS/SYNDIOTACTIC 1,2 STRUCTURE FROM STEREOSPECIFIC POLYMERIZATION VERSALIS SPA (IT) 2021-12-29 EP disclosed
EP-3066139-B1 STEREOREGULAR DIBLOCK POLYBUTADIENES HAVING A 1,4-CIS/SYNDIOTACTIC 1,2 STRUCTURE FROM STEREOSPECIFIC POLYMERIZATION VERSALIS SPA (IT) 2019-02-20 EP disclosed
EP-3394121-A1 PROCESS FOR THE PREPARATION OF (CO) POLYMERS OF CONJUGATED DIENES IN THE PRESENCE OF A CATALYTIC SYSTEM COMPRISING A VANADIUM BIS-IMINE COMPLEX Versalis S.p.A. (IT) 2018-10-31 EP disclosed
US-10093763-B2 Stereoregular diblock polybutadienes having a 1,4-cis/syndiotactic 1,2 structure from stereospecific polymerization VERSALIS S.P.A. (IT) 2018-10-09 US disclosed
US-10066044-B2 Stereoregular diblock polybutadienes having a 1,4-cis/syndiotactic 1,2 structure from stereospecific polymerization VERSALIS S.P.A. (IT) 2018-09-04 US disclosed
WO-2017109767-A1 PROCESS FOR THE PREPARATION OF (CO) POLYMERS OF CONJUGATED DIENES IN THE PRESENCE OF A CATALYTIC SYSTEM COMPRISING A VANADIUM BIS-IMINE COMPLEX VERSALIS S.P.A. (IT) 2017-06-29 WO disclosed
EP-3155686-A1 ELECTROLYTE, CELL AND BATTERY COMPRISING THE ELECTROLYTE, AND USE OF THE ELECTROLYTE Karlsruher Institut Für Technologie (KIT) (DE) 2017-04-19 EP disclosed
WO-1998009999-A2 ALPHA-OLEFIN/VINYLIDENE AROMATIC MONOMER AND/OR HINDERED ALIPHATIC OR CYCLOALIPHATIC VINYLIDENE MONOMER INTERPOLYMERS THE DOW CHEMICAL COMPANY (US) 1998-03-12 WO disclosed
WO-1998010018-A1 BLENDS OF α-OLEFIN/VINYLIDENE AROMATIC MONOMER AND/OR HINDERED ALIPHATIC OR CYCLOALIPHATIC VINYLIDENE MONOMER INTERPOLYMERS THE DOW CHEMICAL COMPANY (US) 1998-03-12 WO disclosed
WO-1998002469-A1 SYNDIOTACTIC/ATACTIC BLOCK POLYOLEFINS, CATALYSTS AND PROCESSES FOR PRODUCING THE SAME FINA RESEARCH S.A. (BE) 1998-01-22 WO disclosed
WO-1997044371-A1 POLYOLEFIN COMPOSITION WITH MOLECULAR WEIGHT MAXIMUM OCCURING IN THAT PART OF THE COMPOSITION THAT HAS THE HIGHEST COMONOMER CONTENT THE DOW CHEMICAL COMPANY (US) 1997-11-27 WO disclosed
WO-1997034943-A1 THERMOPLASTIC ELASTOMERIC CARBON MONOXIDE/OLEFIN COPOLYMERS BASF AKTIENGESELLSCHAFT (DE) 1997-09-25 WO disclosed
WO-1997031029-A1 PROCESS FOR PRODUCING POLYMERS OF ALKENES BY SUSPENSION POLYMERISATION BASF AKTIENGESELLSCHAFT (DE) 1997-08-28 WO disclosed
WO-1997021742-A1 PROCESS FOR THE PREPARATION OF POLYMERISATES OF VINYL AROMATIC COMPOUNDS IN A STAGE USING DOUBLE SCREW EXTRUDERS BASF AKTIENGESELLSCHAFT (DE) 1997-06-19 WO disclosed
WO-1997010286-A1 PROPENE/BUT-1-ENE COPOLYMERS BASF AKTIENGESELLSCHAFT (DE) 1997-03-20 WO disclosed