SCHEMBL4573172

SCHEMBL4573172

CC(C)(C#N)c1ccc(N2CCNCC2)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB1 P08588 9/20 0.53
HTR3E A5X5Y0 4/20 0.49
HTR3B O95264 4/20 0.49
HTR3A P46098 4/20 0.49
HTR3D Q70Z44 4/20 0.49
HTR3C Q8WXA8 4/20 0.49
SIGMAR1 Q99720 4/20 0.49
DRD2 P14416 1/20 0.45
DRD3 P35462 1/20 0.45
ADRB2 P07550 1/20 0.44
NCF1 P14598 1/20 0.44
PLD1 Q13393 1/20 0.44
LTA4H P09960 3/20 0.42
ALDH1A1 P00352 3/20 0.42
KDM4E B2RXH2 1/20 0.42
LMNA P02545 1/20 0.42
SIRT6 Q8N6T7 1/20 0.42
TRPV4 Q9HBA0 1/20 0.41
USP2 O75604 1/20 0.41
TSHR P16473 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL270283 0.80 ADRB1 (0.62) ADRB1HTR3EHTR3BHTR3AHTR3D
SCHEMBL23257306 0.78 ADRB1 (0.55) ADRB1HTR3EHTR3BHTR3AHTR3D
SCHEMBL12088780 0.77 ADRB1 (0.58) ADRB1HTR3EHTR3BHTR3AHTR3D
SCHEMBL4573103 0.77 ADRB1 (0.58) ADRB1HTR3EHTR3BHTR3AHTR3D
SCHEMBL4573136 0.77 PANK3 (0.44) ADRB1PLD1ALDH1A1
SCHEMBL22800963 0.76 CXCR4 (0.53) SIGMAR1ALDH1A1KDM4EUSP2
SCHEMBL8105084 0.76 ALDH1A1 (0.47) ADRB1HTR3EHTR3BHTR3AHTR3D
Hydrochloric Acid SCHEMBL29978981 0.76 PANK3 (0.43) ADRB1ADRB2PLD1ALDH1A1
SCHEMBL4573471 0.76 ADRB1 (0.56) ADRB1HTR3EHTR3BHTR3AHTR3D
Hydrochloric Acid SCHEMBL28880753 0.76 PANK3 (0.43) ADRB1ADRB2PLD1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009001127-A1 CYANOCYCLOPROPYLCARBOXAMIDES AS CATHEPSIN INHIBITORS ASTRAZENECA AB (SE) 2008-12-31 WO disclosed
WO-2009001127-A1 CYANOCYCLOPROPYLCARBOXAMIDES AS CATHEPSIN INHIBITORS ASTRAZENECA AB (SE) 2008-12-31 WO disclosed