SCHEMBL4573265

SCHEMBL4573265

C=CCC(=O)N(Cc1ccc(OC)cc1)[C@H](CC=C)C(=O)OC

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
HTT P42858 2/20 0.41
APLNR P35414 1/20 0.41
BCL2A1 Q16548 4/20 0.40
TDP1 Q9NUW8 1/20 0.39
TP53 P04637 1/20 0.39
CYP3A4 P08684 1/20 0.39
ALOX15 P16050 1/20 0.39
TSHR P16473 1/20 0.39
ALOX12 P18054 1/20 0.39
PSEN1 P49768 1/20 0.39
PSEN2 P49810 1/20 0.39
APH1B Q8WW43 1/20 0.39
NCSTN Q92542 1/20 0.39
APH1A Q96BI3 1/20 0.39
PSENEN Q9NZ42 1/20 0.39
BCHE P06276 1/20 0.39
ACHE P22303 1/20 0.39
YAP1 P46937 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4573275 1.00 ALDH1A1 (0.41) ALDH1A1SMN1; SMN2HTTAPLNRBCL2A1
SCHEMBL25252107 0.74 SMN1; SMN2 (0.57) ALDH1A1SMN1; SMN2HTTBCL2A1TDP1
SCHEMBL13396259 0.74 SMN1; SMN2 (0.57) ALDH1A1SMN1; SMN2HTTBCL2A1TDP1
SCHEMBL19284750 0.72 APLNR (0.54) APLNR
SCHEMBL19284814 0.72 APLNR (0.54) APLNR
SCHEMBL19284751 0.72 APLNR (0.54) APLNR
SCHEMBL20447205 0.72 ALDH1A1 (0.54) ALDH1A1SMN1; SMN2HTTBCL2A1TDP1
SCHEMBL15209869 0.72 APLNR (0.44) ALDH1A1SMN1; SMN2HTTAPLNRBCL2A1
SCHEMBL15209867 0.72 APLNR (0.44) ALDH1A1SMN1; SMN2HTTAPLNRBCL2A1
SCHEMBL8922383 0.71 ATM (0.43) ALDH1A1SMN1; SMN2HTTTDP1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008031788-A1 AMINOAZEPINE DERIVATIVES AS HIGHLY EFFICIENT INHIBITORS OF THE INDUCIBLE NITRIC OXIDE SYNTHASE NYCOMED GMBH (DE) 2008-03-20 WO disclosed
WO-2008031788-A1 AMINOAZEPINE DERIVATIVES AS HIGHLY EFFICIENT INHIBITORS OF THE INDUCIBLE NITRIC OXIDE SYNTHASE NYCOMED GMBH (DE) 2008-03-20 WO disclosed