SCHEMBL4573344

SCHEMBL4573344

CC(=O)ON=CCc1ccc(Br)cc1O

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 7/20 0.38
KMT2A Q03164 5/20 0.38
KDM4E B2RXH2 4/20 0.38
POLB P06746 2/20 0.38
GAA P10253 4/20 0.36
HPGD P15428 3/20 0.36
HTT P42858 3/20 0.36
SMN1; SMN2 Q16637 1/20 0.34
CES2 O00748 1/20 0.33
GALR3 O60755 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2C9 P11712 1/20 0.33
ALOX15 P16050 1/20 0.33
CASP1 P29466 1/20 0.33
CYP2C19 P33261 1/20 0.33
UCHL1 P09936 1/20 0.33
UCHL3 P15374 1/20 0.33
MAOA P21397 3/20 0.33
MAOB P27338 3/20 0.33
NPSR1 Q6W5P4 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4573203 0.75 ALOX15 (0.38) MAPTKMT2AKDM4EPOLBGAA
SCHEMBL2144792 0.75 ALOX15 (0.38) MAPTKMT2AKDM4EPOLBGAA
SCHEMBL1897113 0.71 ERN1 (0.47) HPGDHTTCES2GALR3CYP1A2
SCHEMBL9900604 0.71 THRB (0.37) MAPTKMT2AKDM4EPOLBHPGD
SCHEMBL9900406 0.70 PTPN1 (0.41) MAPTKDM4EPOLBGAACASP1
SCHEMBL15658116 0.70 MAPT (0.46) MAPTPOLBGAAHPGDCES2
SCHEMBL30777878 0.69 ALOX15 (0.44) KDM4EPOLBGAAHPGDHTT
SCHEMBL1005997 0.69 ALOX15 (0.44) KDM4EPOLBGAAHPGDHTT
SCHEMBL2450978 0.68 HTT (0.36) KMT2AHPGDHTTCYP2C9CYP2C19
SCHEMBL472482 0.68 GABRA1 (0.50) MAPTKMT2AKDM4EPOLBGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009001127-A1 CYANOCYCLOPROPYLCARBOXAMIDES AS CATHEPSIN INHIBITORS ASTRAZENECA AB (SE) 2008-12-31 WO disclosed