SCHEMBL4580599

SCHEMBL4580599

COc1cc(OC(=O)c2cccs2)ccc1-c1ccc2c(c1C(N)c1ccccc1OC)N(C)C(=O)C(C)(C)N2

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IL6 P05231 8/20 0.41
PLA2G1B P04054 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
ATG4B Q9Y4P1 1/20 0.37
ALDH1A1 P00352 5/20 0.36
MAPT P10636 4/20 0.36
HPGD P15428 2/20 0.36
LMNA P02545 1/20 0.36
CYP1A1 P04798 1/20 0.35
CYP1B1 Q16678 1/20 0.35
C1S P09871 2/20 0.35
CFD P00746 1/20 0.35
HDAC6 Q9UBN7 1/20 0.35
KMT2A Q03164 4/20 0.35
KDM4E B2RXH2 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2C19 P33261 1/20 0.35
POLB P06746 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4129531 0.88 IL6 (0.41) IL6ALDH1A1KDM4E
SCHEMBL4140035 0.85 IL6 (0.42) IL6
SCHEMBL4142446 0.84 LMNA (0.46) IL6TDP1ALDH1A1MAPTLMNA
SCHEMBL13571452 0.83 IL6 (0.41) IL6PLA2G1BTDP1ATG4BALDH1A1
SCHEMBL4580605 0.81 IL6 (0.46) IL6TDP1ALDH1A1MAPTHPGD
SCHEMBL1315415 0.81 NR3C1 (0.42) PLA2G1BTDP1ATG4BALDH1A1MAPT
SCHEMBL4581403 0.80 IL6 (0.51) IL6TDP1ALDH1A1MAPTLMNA
SCHEMBL4581832 0.79 ACHE (0.41) IL6TDP1ALDH1A1MAPTLMNA
SCHEMBL6114280 0.79 IL6 (0.42) IL6TDP1ALDH1A1MAPTHPGD
SCHEMBL14015605 0.79 KMT2A (0.36) IL6PLA2G1BTDP1ATG4BALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1995242-A1 NOVEL 1,2,3,4-TETRAHYDROQUINOXALINE DERIVATIVE HAVING GLUCOCORTICOID RECEPTOR BINDING ACTIVITY Santen Pharmaceutical Co., Ltd (JP) 2008-11-26 EP disclosed