SCHEMBL458229

SCHEMBL458229

N#Cc1ccc(Oc2ccc(C(F)(F)F)cc2)cc1

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 2/20 0.68
PARP15 Q460N3 1/20 0.49
PARP10 Q53GL7 1/20 0.49
PARP2 Q9UGN5 1/20 0.49
LTA4H P09960 2/20 0.48
CYP19A1 P11511 3/20 0.47
KDM4E B2RXH2 2/20 0.47
LMNA P02545 2/20 0.47
MEN1 O00255 1/20 0.47
POLB P06746 1/20 0.47
MAPT P10636 1/20 0.47
PKM P14618 1/20 0.47
MAPK1 P28482 1/20 0.47
RAB9A P51151 1/20 0.47
KMT2A Q03164 1/20 0.47
IL18 Q14116 1/20 0.47
CYP3A4 P08684 1/20 0.46
CYP3A5 P20815 1/20 0.46
EPHX2 P34913 1/20 0.44
SCN8A Q9UQD0 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL524351 0.87 KIF11 (0.86) KIF11CYP19A1KDM4EMEN1KMT2A
Hydrochloric Acid SCHEMBL27812058 0.85 KIF11 (0.83) KIF11CYP19A1KDM4EMEN1KMT2A
SCHEMBL11148692 0.82 CA1 (0.52) KIF11LTA4HMAPTMAPK1RAB9A
SCHEMBL1685383 0.82 CA1 (0.52) KIF11LTA4HMAPTMAPK1RAB9A
SCHEMBL7041250 0.82 PARP15 (0.63) PARP15PARP10PARP2CYP19A1KDM4E
SCHEMBL8852392 0.82 PARP15 (0.63) PARP15PARP10PARP2CYP19A1KDM4E
SCHEMBL16626137 0.81 KIF11 (0.76) KIF11CYP19A1KDM4EMEN1KMT2A
SCHEMBL3456838 0.81 KIF11 (1.00) KIF11CYP19A1CYP3A4CYP3A5PTPN5
SCHEMBL13063632 0.81 KIF11 (1.00) KIF11CYP19A1CYP3A4CYP3A5PTPN5
SCHEMBL10710562 0.80 KIF11 (0.58) KIF11PARP15PARP10PARP2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-3954829-A HERBICIDES BAYER AKTIENGESELLSCHAFT (DT) 1976-05-04 US claimed
US-9045442-B2 Antibacterial compounds and methods of using same UNIVERSITY OF NOTRE DAME DU LAC (US) 2015-06-02 US disclosed
WO-2012032261-A1 METHOD FOR SYNTHESISING BIARYL ETHER OR BIHETEROARYL ETHER CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (C.N.R.S) (FR) 2012-03-15 WO disclosed
WO-2011078370-A1 NOVEL PARABANIC ACID DERIVATIVE AND DRUG HAVING THE SAME AS ACTIVE INGREDIENT 杏林製薬株式会社 (JP) 2011-06-30 WO disclosed
US-20100261673-A1 ANTIBACTERIAL COMPOUNDS AND METHODS OF USING SAME UNIVERSITY OF NOTRE DAME DU LAC (US) 2010-10-14 US disclosed
WO-2009082398-A1 ANTIBACTERIAL COMPOUNDS AND METHODS OF USING SAME UNIVERSITY OF NOTRE DAME DU LAC (US) 2009-07-02 WO disclosed
WO-2009041972-A1 ANTIBACTERIAL COMPOUNDS AND METHODS OF USING SAME UNIVERSITY OF NOTRE DAME DU LAC (US) 2009-04-02 WO disclosed
US-3954829-A HERBICIDES BAYER AKTIENGESELLSCHAFT (DT) 1976-05-04 US disclosed
US-3954829-A HERBICIDES BAYER AKTIENGESELLSCHAFT (DT) 1976-05-04 US disclosed
US-3954829-A HERBICIDES BAYER AKTIENGESELLSCHAFT (DT) 1976-05-04 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100261673-A1 ANTIBACTERIAL COMPOUNDS AND METHODS OF USING SAME SPOUT1, MRPL21, NPEPPS KIF11 3772/4885PARP15 192/4885PARP10 231/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.