SCHEMBL4585487

SCHEMBL4585487

CC(N)CCN1CCC(N(Cc2ccsc2)c2cccnc2)CC1

nearest known ligand 0.41

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 7/20 0.41
OPRD1 P41143 7/20 0.41
OPRK1 P41145 7/20 0.41
CCR5 P51681 3/20 0.38
KDM4E B2RXH2 1/20 0.38
ALDH1A1 P00352 1/20 0.38
CYP3A4 P08684 4/20 0.37
DRD2 P14416 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4244588 0.83 CCR5 (0.46) CCR5
SCHEMBL4586423 0.82 CCR5 (0.41) OPRM1OPRD1OPRK1CCR5DRD2
SCHEMBL4585402 0.81 CCR5 (0.41) OPRM1OPRD1OPRK1CCR5KDM4E
SCHEMBL4585393 0.81 CCR5 (0.53) OPRM1OPRD1OPRK1CCR5
SCHEMBL4587616 0.80 CCR5 (0.42) OPRM1OPRD1OPRK1CCR5DRD2
SCHEMBL4244585 0.79 CCR5 (0.46) CCR5CYP3A4
SCHEMBL4585491 0.78 CCR5 (0.44) OPRM1OPRD1OPRK1CCR5ALDH1A1
SCHEMBL5056837 0.77 CCR5 (0.51) OPRM1CCR5KDM4EALDH1A1CYP3A4
SCHEMBL5057871 0.77 CCR5 (0.44) CCR5KDM4EALDH1A1CYP3A4
SCHEMBL5056393 0.74 CCR5 (0.49) OPRM1CCR5CYP3A4DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1708703-A4 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC (CA) 2008-04-09 EP disclosed
EP-1708703-A2 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC. (CA) 2006-10-11 EP disclosed
WO-2005059107-A2 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC. (CA) 2005-06-30 WO disclosed