SCHEMBL4586423

SCHEMBL4586423

C[C@@H](N)CCN1CCC(N(Cc2ccsc2)c2ccc(F)cc2)CC1

nearest known ligand 0.41

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 6/20 0.41
OPRM1 P35372 8/20 0.39
OPRD1 P41143 6/20 0.39
OPRK1 P41145 6/20 0.39
CCR2 P41597 1/20 0.36
TMEM97 Q5BJF2 1/20 0.36
HRH3 Q9Y5N1 1/20 0.35
DRD2 P14416 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4585393 0.88 CCR5 (0.53) CCR5OPRM1OPRD1OPRK1
SCHEMBL4585402 0.88 CCR5 (0.41) CCR5OPRM1OPRD1OPRK1DRD2
SCHEMBL4587616 0.87 CCR5 (0.42) CCR5OPRM1OPRD1OPRK1DRD2
SCHEMBL4585491 0.87 CCR5 (0.44) CCR5OPRM1OPRD1OPRK1
SCHEMBL4585487 0.82 OPRM1 (0.41) CCR5OPRM1OPRD1OPRK1DRD2
SCHEMBL4239765 0.82 CCR5 (0.51) CCR5
SCHEMBL4243416 0.77 CCR5 (0.51) CCR5OPRM1
SCHEMBL4586437 0.75 CCR5 (0.47) CCR5OPRM1TMEM97
SCHEMBL4586731 0.73 OPRM1 (0.53) CCR5OPRM1DRD2
SCHEMBL4586432 0.71 CCR5 (0.54) CCR5DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1708703-A4 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC (CA) 2008-04-09 EP disclosed
EP-1708703-A2 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC. (CA) 2006-10-11 EP disclosed
WO-2005059107-A2 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC. (CA) 2005-06-30 WO disclosed