SCHEMBL4585402

SCHEMBL4585402

CSc1ccc(N(Cc2ccsc2)C2CCN(CC[C@@H](C)N)CC2)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 3/20 0.41
OPRM1 P35372 9/20 0.38
OPRD1 P41143 8/20 0.38
OPRK1 P41145 8/20 0.38
SLC6A2 P23975 2/20 0.34
SLC6A4 P31645 2/20 0.34
SLC6A3 Q01959 2/20 0.34
MAOA P21397 1/20 0.34
DRD2 P14416 1/20 0.34
CHRM2 P08172 3/20 0.33
CHRM1 P11229 3/20 0.33
HTR1A P08908 1/20 0.33
ADRA2A P08913 1/20 0.33
DRD1 P21728 1/20 0.33
ADRA1A P35348 1/20 0.33
DRD3 P35462 1/20 0.33
KCNH2 Q12809 1/20 0.33
CHRM3 P20309 2/20 0.33
HTR1D P28221 1/20 0.33
HTR1B P28222 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4586423 0.88 CCR5 (0.41) CCR5OPRM1OPRD1OPRK1DRD2
SCHEMBL4585393 0.86 CCR5 (0.53) CCR5OPRM1OPRD1OPRK1
SCHEMBL4587616 0.85 CCR5 (0.42) CCR5OPRM1OPRD1OPRK1SLC6A2
SCHEMBL4585491 0.83 CCR5 (0.44) CCR5OPRM1OPRD1OPRK1SLC6A4
SCHEMBL4241214 0.82 CCR5 (0.49) CCR5KCNH2
SCHEMBL4585487 0.81 OPRM1 (0.41) CCR5OPRM1OPRD1OPRK1DRD2
SCHEMBL4245513 0.78 CCR5 (0.49) CCR5KCNH2
SCHEMBL4586731 0.71 OPRM1 (0.53) CCR5OPRM1DRD2CHRM2CHRM3
SCHEMBL13931614 0.70 CCR5 (0.81) CCR5KCNH2
SCHEMBL4240431 0.70 CCR5 (0.53) CCR5KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1708703-A4 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC (CA) 2008-04-09 EP disclosed
EP-1708703-A2 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC. (CA) 2006-10-11 EP disclosed
WO-2005059107-A2 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC. (CA) 2005-06-30 WO disclosed