SCHEMBL4585393

SCHEMBL4585393

COc1ccc(N(Cc2ccsc2)C2CCN(CC[C@@H](C)N)CC2)cc1

nearest known ligand 0.53

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 8/20 0.53
OPRM1 P35372 8/20 0.43
OPRD1 P41143 5/20 0.43
OPRK1 P41145 5/20 0.43
OPRL1 P41146 1/20 0.39
CTSD P07339 1/20 0.38
FFAR1 O14842 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4585491 0.89 CCR5 (0.44) CCR5OPRM1OPRD1OPRK1
SCHEMBL4586423 0.88 CCR5 (0.41) CCR5OPRM1OPRD1OPRK1
SCHEMBL4585402 0.86 CCR5 (0.41) CCR5OPRM1OPRD1OPRK1
SCHEMBL4586731 0.86 OPRM1 (0.53) CCR5OPRM1
SCHEMBL4587616 0.85 CCR5 (0.42) CCR5OPRM1OPRD1OPRK1OPRL1
SCHEMBL4243511 0.82 CCR5 (0.64) CCR5
SCHEMBL4240067 0.82 CCR5 (0.64) CCR5
SCHEMBL4585487 0.81 OPRM1 (0.41) CCR5OPRM1OPRD1OPRK1
SCHEMBL5056837 0.81 CCR5 (0.51) CCR5OPRM1OPRL1
SCHEMBL4243509 0.78 CCR5 (0.64) CCR5OPRM1OPRD1OPRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1708703-A4 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC (CA) 2008-04-09 EP disclosed
EP-1708703-A2 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC. (CA) 2006-10-11 EP disclosed
WO-2005059107-A2 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC. (CA) 2005-06-30 WO disclosed