SCHEMBL4585491

SCHEMBL4585491

C[C@@H](N)CCN1CCC(N(Cc2ccsc2)c2ccc(OC(F)(F)F)cc2)CC1

nearest known ligand 0.44

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 6/20 0.44
CARM1 Q86X55 1/20 0.37
PRMT6 Q96LA8 1/20 0.37
ALDH1A1 P00352 1/20 0.36
OPRM1 P35372 5/20 0.36
OPRD1 P41143 5/20 0.36
OPRK1 P41145 5/20 0.36
CHRM4 P08173 1/20 0.36
PDK1 Q15118 1/20 0.35
SLC6A4 P31645 2/20 0.35
SLC6A3 Q01959 2/20 0.35
UBE2M P61081 1/20 0.34
DCUN1D1 Q96GG9 1/20 0.34
TSHR P16473 1/20 0.34
HTR2A P28223 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4585393 0.89 CCR5 (0.53) CCR5OPRM1OPRD1OPRK1
SCHEMBL4586423 0.87 CCR5 (0.41) CCR5OPRM1OPRD1OPRK1
SCHEMBL4245439 0.84 CCR5 (0.53) CCR5UBE2MDCUN1D1
SCHEMBL4237093 0.84 CCR5 (0.53) CCR5UBE2MDCUN1D1
SCHEMBL4585402 0.83 CCR5 (0.41) CCR5ALDH1A1OPRM1OPRD1OPRK1
SCHEMBL4587616 0.82 CCR5 (0.42) CCR5OPRM1OPRD1OPRK1SLC6A4
SCHEMBL4237091 0.80 CCR5 (0.52) CCR5PDK1UBE2MDCUN1D1
SCHEMBL4245437 0.80 CCR5 (0.52) CCR5PDK1UBE2MDCUN1D1
SCHEMBL4585487 0.78 OPRM1 (0.41) CCR5ALDH1A1OPRM1OPRD1OPRK1
SCHEMBL4586731 0.75 OPRM1 (0.53) CCR5OPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1708703-A4 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC (CA) 2008-04-09 EP disclosed
EP-1708703-A2 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC. (CA) 2006-10-11 EP disclosed
WO-2005059107-A2 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC. (CA) 2005-06-30 WO disclosed