SCHEMBL4585573

SCHEMBL4585573

CC(=O)Nc1ccc(N(C2CCNCC2)[C@H](C)CCN)cn1

nearest known ligand 0.36

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HTR1F P30939 1/20 0.36
PTK2 Q05397 1/20 0.36
CYP1A2 P05177 1/20 0.34
GAA P10253 1/20 0.34
ABL1 P00519 1/20 0.34
CYP3A4 P08684 1/20 0.34
BCR P11274 1/20 0.34
MKNK1 Q9BUB5 1/20 0.34
MKNK2 Q9HBH9 1/20 0.34
GSK3B P49841 1/20 0.33
DYRK1A Q13627 1/20 0.33
GRIN2B Q13224 2/20 0.33
GLS O94925 1/20 0.32
TLR9 Q9NR96 1/20 0.32
TLR8 Q9NR97 1/20 0.32
TLR7 Q9NYK1 1/20 0.32
PARP1 P09874 1/20 0.32
DHODH Q02127 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4585576 0.80 HTR1F (0.36) HTR1FPTK2CYP1A2GAAABL1
SCHEMBL4585642 0.75 LOXL2 (0.39) GAA
SCHEMBL4001973 0.72 GCK (0.41) ABL1
SCHEMBL3997886 0.71 ALOX15 (0.44) GAACYP3A4
SCHEMBL4001474 0.69 HTR1F (0.37) HTR1FCYP1A2TLR9TLR8TLR7
SCHEMBL4002694 0.69 SLC6A4 (0.39) ABL1
SCHEMBL3997555 0.69 REN (0.40)
SCHEMBL4003258 0.68 SLC6A2 (0.37) HTR1FCYP1A2
SCHEMBL3997842 0.67 PTK2 (0.37) HTR1FPTK2CYP1A2GAA
SCHEMBL3999681 0.67 SLC6A2 (0.36) HTR1FPTK2CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1708703-A4 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC (CA) 2008-04-09 EP disclosed
EP-1708703-A2 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC. (CA) 2006-10-11 EP disclosed
WO-2005059107-A2 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC. (CA) 2005-06-30 WO disclosed