SCHEMBL4586020

SCHEMBL4586020

CC(C)(C)OC(=O)Nc1c(F)cccc1C(=O)N(Cc1ccccc1)C1CCNCC1

nearest known ligand 0.48

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
DCUN1D1 Q96GG9 3/20 0.48
SLC6A2 P23975 6/20 0.42
SLC6A4 P31645 6/20 0.42
SLC6A3 Q01959 5/20 0.41
MAPT P10636 1/20 0.41
AGER Q15109 2/20 0.39
ALDH1A1 P00352 1/20 0.39
MTNR1A P48039 1/20 0.39
TACR1 P25103 2/20 0.39
AKT1 P31749 2/20 0.38
KCNH2 Q12809 2/20 0.38
UBE2M P61081 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5744569 0.86 DCUN1D1 (0.52) DCUN1D1SLC6A2SLC6A4SLC6A3MAPT
SCHEMBL16227662 0.74 TACR1 (0.47) DCUN1D1SLC6A2SLC6A4SLC6A3ALDH1A1
SCHEMBL17870701 0.73 DCUN1D1 (0.51) DCUN1D1SLC6A2SLC6A4SLC6A3MAPT
SCHEMBL1346055 0.72 ALB (0.44) ALDH1A1
SCHEMBL526963 0.70 AGER (0.46) DCUN1D1SLC6A2SLC6A4SLC6A3MAPT
SCHEMBL5042994 0.70 SLC6A2 (0.53) DCUN1D1SLC6A2SLC6A4SLC6A3TACR1
SCHEMBL3811903 0.70 DCUN1D1 (0.58) DCUN1D1SLC6A2SLC6A4SLC6A3AGER
SCHEMBL3601820 0.70 L3MBTL1 (0.60)
SCHEMBL14417236 0.70 SLC6A4 (0.47) SLC6A2SLC6A4SLC6A3TACR1KCNH2
SCHEMBL3837699 0.70 SLC6A2 (0.49) DCUN1D1SLC6A2SLC6A4SLC6A3AKT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1689493-A4 CALCITONIN GENE RELATED PEPTIDE RECEPTOR ANTAGONISTS BRISTOL MYERS SQUIBB CO (US) 2008-04-23 EP disclosed
EP-1689738-A2 HETEROCYCLIC ANTI-MIGRAINE AGENTS Bristol-Myers Squibb Company (US) 2006-08-16 EP disclosed
EP-1689493-A1 CALCITONIN GENE RELATED PEPTIDE RECEPTOR ANTAGONISTS Bristol-Myers Squibb Pharma Company (US) 2006-08-16 EP disclosed
WO-2005065779-A1 CALCITONIN GENE RELATED PEPTIDE RECEPTOR ANTAGONISTS BRISTOL-MYERS SQUIBB COMPANY (US) 2005-07-21 WO disclosed
WO-2005056550-A2 HETEROCYCLIC ANTI-MIGRAINE AGENTS BRISTOL-MYERS SQUIBB COMPANY (US) 2005-06-23 WO disclosed